SCHEMBL4958574

SCHEMBL4958574

COc1ccc(C(COC(N)=O)c2nnn[nH]2)c(OC)c1OC

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.38
AOC3 Q16853 2/20 0.38
CYP1A2 P05177 2/20 0.38
LMNA P02545 2/20 0.38
KDM4E B2RXH2 2/20 0.38
PDE4D Q08499 1/20 0.33
PKM P14618 2/20 0.33
CYP2D6 P10635 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
MAPT P10636 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
MAPK1 P28482 1/20 0.32
DPP4 P27487 1/20 0.31
PDK1 Q15118 1/20 0.31
LDHA P00338 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4958548 0.74 CES2 (0.35) SMN1; SMN2CYP1A2PKMCYP2D6NPSR1
SCHEMBL4959933 0.74 CYP1A2 (0.41) SMN1; SMN2CYP1A2LMNAKDM4EPKM
SCHEMBL4962125 0.74 CYP1A2 (0.41) SMN1; SMN2CYP1A2LMNAKDM4EPKM
SCHEMBL4959934 0.72 CYP1A2 (0.38) SMN1; SMN2CYP1A2PKMCYP2D6NPSR1
SCHEMBL4958729 0.71 SMN1; SMN2 (0.38) SMN1; SMN2CYP1A2PKMCYP2D6NPSR1
SCHEMBL4960360 0.70 CYP1A2 (0.33) SMN1; SMN2CYP1A2PKMCYP2D6NPSR1
SCHEMBL4960105 0.68 SMN1; SMN2 (0.43) SMN1; SMN2CYP1A2PKMCYP2D6NPSR1
SCHEMBL4960423 0.68 CYP1A2 (0.38) SMN1; SMN2CYP1A2KDM4EPKMCYP2D6
SCHEMBL4962975 0.65 ALOX5 (0.46) LMNAHTT
SCHEMBL16793190 0.64 AOC3 (0.49) SMN1; SMN2AOC3CYP1A2LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879873-A1 NEUROTHERAPEUTIC AZOLE COMPOUNDS SK Holdings Co., Ltd. (KR) 2008-01-23 EP disclosed
WO-2006112685-A1 NEUROTHERAPEUTIC AZOLE COMPOUNDS SK HOLDINGS CO., LTD. (KR) 2006-10-26 WO disclosed