SCHEMBL4959467

SCHEMBL4959467

COCCCN1CCOc2ccc(CO[C@H]3CN(S(=O)(=O)c4ccc(C)cc4)[C@H](CO)C[C@@H]3c3ccc(COC)cc3)cc21

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.36
KMT2A Q03164 4/20 0.34
REN P00797 1/20 0.33
POLB P06746 2/20 0.33
MEN1 O00255 1/20 0.32
MAPT P10636 2/20 0.31
THRB P10828 1/20 0.31
LMNA P02545 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
RORC P51449 3/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1036293 0.95 CYP2C9 (0.35) CYP2C9KMT2ARENPOLBMEN1
SCHEMBL2920405 0.95 FKBP1A (0.36) CYP2C9KMT2AMAPTLMNASMN1; SMN2
SCHEMBL4961309 0.93 CYP2C9 (0.35) CYP2C9KMT2ARENPOLBMEN1
SCHEMBL1517806 0.93 CYP2C9 (0.33) CYP2C9KMT2ARENPOLBLMNA
SCHEMBL1517808 0.93 CYP2C9 (0.33) CYP2C9KMT2ARENPOLBLMNA
SCHEMBL4959427 0.91 CYP2C9 (0.35) CYP2C9KMT2ARENPOLBMEN1
SCHEMBL2390330 0.90 CYP2C9 (0.32) CYP2C9KMT2ARENRORC
SCHEMBL2390336 0.90 CYP2C9 (0.32) CYP2C9KMT2ARENRORC
SCHEMBL2922224 0.90 CYP2C9 (0.34) CYP2C9KMT2ARENPOLBMEN1
SCHEMBL2916824 0.90 FKBP1A (0.35) CYP2C9KMT2AMAPTLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1897879-A2 2,4,5 substituted piperidines as renin inhibitors Speedel Experimenta AG (CH) 2008-03-12 EP disclosed