SCHEMBL4962973

SCHEMBL4962973

COC(=O)NCCCc1cccc([N+](=O)[O-])c1O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 1/20 0.45
PTPN1 P18031 2/20 0.44
KMT2A Q03164 3/20 0.42
ALDH1A1 P00352 1/20 0.41
HTT P42858 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
POLB P06746 1/20 0.41
CYP2C19 P33261 1/20 0.41
CRHBP P24387 2/20 0.40
CRHR2 Q13324 2/20 0.40
MTNR1A P48039 2/20 0.40
G6PD P11413 1/20 0.40
MTNR1B P49286 1/20 0.40
MEN1 O00255 2/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
MGLL Q99685 1/20 0.40
KDM4E B2RXH2 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2016391 0.78 GPR35 (0.56) GPR35ALDH1A1CYP2C19
SCHEMBL4099366 0.77 TDP1 (0.50) PTPN1KMT2AALDH1A1L3MBTL1POLB
SCHEMBL4101146 0.77 PTPN1 (0.46) PTPN1KMT2AALDH1A1HTTL3MBTL1
SCHEMBL8326737 0.77 CYP4A11 (0.50) GPR35PTPN1KMT2AALDH1A1HTT
SCHEMBL8402772 0.75 GPR35 (0.53) GPR35KDM4E
SCHEMBL10267923 0.75 GPR35 (0.53) GPR35PTPN1KMT2AALDH1A1L3MBTL1
SCHEMBL27864868 0.75 GPR35 (0.53) GPR35KMT2AALDH1A1L3MBTL1MEN1
SCHEMBL5595098 0.74 GPR35 (0.60) GPR35KMT2AALDH1A1POLBCYP2C19
SCHEMBL20495063 0.74 MEN1 (0.59) PTPN1KMT2AALDH1A1HTTL3MBTL1
SCHEMBL27648916 0.74 GPR35 (0.55) GPR35KMT2AALDH1A1HTTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879858-A2 PROCESSES FOR PREPARING BIARYL UREAS AND ANALOGS THEREOF Vertex Pharmaceuticals, Inc. (US) 2008-01-23 EP disclosed
WO-2006122072-A2 PROCESSES FOR PREPARING BIARYL UREAS AND ANALOGS THEREOF VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-11-16 WO disclosed