SCHEMBL496340

SCHEMBL496340

Cc1c([N+](=O)[O-])cc([N+](=O)[O-])c(C(C)(C(=O)O)C(=O)O)c1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 3/20 0.40
TSHR P16473 5/20 0.36
ALDH1A1 P00352 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP1A2 P05177 2/20 0.36
HPGD P15428 1/20 0.36
ALOX15 P16050 1/20 0.36
HIF1A Q16665 1/20 0.36
TXNRD1 Q16881 1/20 0.36
TXNRD3 Q86VQ6 1/20 0.36
TXNRD2 Q9NNW7 1/20 0.36
THRB P10828 1/20 0.35
LMNA P02545 1/20 0.35
CYP2D6 P10635 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3304363 0.70 TSHR (0.57) GPR35TSHRALDH1A1TDP1CYP3A4
SCHEMBL4595029 0.69 TSHR (0.50) GPR35TSHRALDH1A1TDP1CYP3A4
SCHEMBL29029703 0.69 ALDH1A1 (0.42) GPR35TSHRALDH1A1TDP1CYP3A4
SCHEMBL2098784 0.68 GPR35 (0.57) GPR35TSHRALDH1A1TDP1CYP3A4
SCHEMBL3536339 0.68 TSHR (0.45) TSHRALDH1A1TDP1CYP3A4LMNA
SCHEMBL11852169 0.68 MAPK1 (0.50) GPR35TSHRALDH1A1TDP1CYP3A4
SCHEMBL11852183 0.68 MAPK1 (0.50) GPR35TSHRALDH1A1TDP1CYP3A4
SCHEMBL11758012 0.68 TDP1 (0.55) GPR35TSHRTDP1CYP1A2LMNA
SCHEMBL8658889 0.68 CYP1A2 (0.55) GPR35TSHRALDH1A1TDP1CYP3A4
SCHEMBL10614473 0.67 GPR35 (0.53) GPR35TSHRALDH1A1TDP1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106190-B2 2-aminobenzamide derivatives ASTELLAS PHARMA INC. (JP) 2012-01-31 US disclosed