SCHEMBL4964264

SCHEMBL4964264

CCCCCCCN(Cc1ccc(F)cc1F)C(=O)COc1ccc(CCOc2c(C)cccc2C(=O)O)cc1OC

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LPAR1 Q92633 6/20 0.41
PPARG P37231 1/20 0.40
PPARA Q07869 1/20 0.40
BCHE P06276 3/20 0.38
LPAR5 Q9H1C0 2/20 0.37
HTR2A P28223 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4961660 0.91 PPARG (0.45) KDM4EALDH1A1LPAR1PPARGPPARA
SCHEMBL4961998 0.86 KDM4E (0.43) KDM4EALDH1A1HTR2A
SCHEMBL4964263 0.85 HSP90AA1 (0.44) KDM4EALDH1A1
SCHEMBL4961989 0.83 ALDH1A1 (0.50) KDM4EALDH1A1PPARGPPARAHTR2A
SCHEMBL4964280 0.82 KDM4E (0.46) KDM4EALDH1A1LPAR1PPARGPPARA
SCHEMBL4964260 0.77 KDM4E (0.39) KDM4EALDH1A1LPAR1PPARGPPARA
SCHEMBL4965190 0.73 HTR2A (0.43) ALDH1A1LPAR1LPAR5HTR2A
SCHEMBL4630408 0.70 LTB4R2 (0.48) PPARGPPARAHTR2A
SCHEMBL4629932 0.70 HTR2A (0.49) LPAR1PPARGPPARALPAR5HTR2A
SCHEMBL4963240 0.69 PPARD (0.44) LPAR1PPARGPPARALPAR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1517679-B1 ORTHO-SUBSTITUTED BENZOIC ACID DERIVATIVES FOR THE TREATMENT OF INSULIN RESISTANCE ASTRAZENECA AB (SE) 2008-02-13 EP disclosed