SCHEMBL4964541

SCHEMBL4964541

COC(Br)(Cc1ccccc1)OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.50
TAAR1 Q96RJ0 1/20 0.50
CYP2D6 P10635 2/20 0.46
LMNA P02545 1/20 0.46
CYP1A2 P05177 3/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
TRPA1 O75762 2/20 0.42
TSHR P16473 2/20 0.42
TP53 P04637 1/20 0.42
ALDH1A1 P00352 1/20 0.42
LTA4H P09960 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
HIF1A Q16665 1/20 0.40
CALM1 P0DP23 1/20 0.39
FDPS P14324 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CYP1A1 P04798 1/20 0.38
CYP1B1 Q16678 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6909686 0.80 SLC6A2 (0.50) SLC6A2TAAR1CYP2D6LMNACYP1A2
SCHEMBL5088767 0.80 SLC6A2 (0.50) SLC6A2TAAR1CYP2D6LMNACYP1A2
SCHEMBL6551711 0.79 SLC6A2 (0.50) SLC6A2TAAR1CYP2D6LMNACYP1A2
SCHEMBL10462120 0.78 SLC6A2 (0.54) SLC6A2TAAR1CYP2D6LMNACYP1A2
SCHEMBL872871 0.78 SLC6A2 (0.54) SLC6A2TAAR1CYP2D6LMNACYP1A2
SCHEMBL25407758 0.76 TAAR1 (0.58) SLC6A2TAAR1CYP2D6LMNACYP1A2
SCHEMBL828471 0.76 TAAR1 (0.58) SLC6A2TAAR1CYP2D6LMNACYP1A2
SCHEMBL9776240 0.76 SLC6A2 (0.46) SLC6A2TAAR1CYP2D6LMNACYP1A2
SCHEMBL9862386 0.76 CYP1A2 (0.50) SLC6A2TAAR1CYP2D6LMNACYP1A2
SCHEMBL940763 0.76 SLC6A2 (0.46) SLC6A2TAAR1CYP2D6LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1885704-A2 ANTAGONISTS OF THE VANILLOID RECEPTOR SUBTYPE 1 (VR1) AND USES THEREOF Abbott Laboratories (US) 2008-02-13 EP disclosed
WO-2006135383-A2 INDAZOLES MYRIAD GENETICS, INC. (US) 2006-12-21 WO disclosed
WO-2006122250-A2 ANTAGONISTS OF THE VANILLOID RECEPTOR SUBTYPE 1 (VR1) AND USES THEREOF ABBOTT LABORATORIES (US) 2006-11-16 WO disclosed
EP-1218376-A4 TYROSINE KINASE INHIBITORS MERCK & CO INC (US) 2002-11-20 EP disclosed
EP-1218376-A1 TYROSINE KINASE INHIBITORS Merck & Co., Inc. (US) 2002-07-03 EP disclosed
WO-2001017995-A1 TYROSINE KINASE INHIBITORS MERCK & CO., INC. (US) 2001-03-15 WO disclosed