SCHEMBL4964876

SCHEMBL4964876

CS(=O)(=O)Oc1c(-c2cccc(F)c2)nc2ccccc2c1C(=O)NCCCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 15/20 0.51
LMNA P02545 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.44
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4962172 0.97 TACR3 (0.50) TACR3LMNAL3MBTL1
SCHEMBL4961957 0.95 TACR3 (0.51) TACR3LMNAL3MBTL1
SCHEMBL4963091 0.91 LMNA (0.60) TACR3LMNAL3MBTL1
SCHEMBL4963863 0.83 LMNA (0.54) TACR3LMNAL3MBTL1
SCHEMBL4962076 0.81 LMNA (0.57) TACR3LMNAL3MBTL1
SCHEMBL4961927 0.81 LMNA (0.52) TACR3LMNAL3MBTL1NPC1RAB9A
SCHEMBL4963768 0.80 LMNA (0.52) TACR3LMNAL3MBTL1NPC1RAB9A
SCHEMBL4967704 0.79 TACR3 (0.74) TACR3
SCHEMBL4966074 0.79 TACR3 (0.74) TACR3
SCHEMBL4965436 0.78 TACR3 (0.70) TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1896418-A1 QUINOLINE 3 -SULFONATE ESTERS AS NK3 RECEPTOR MODULATORS AstraZeneca AB (SE) 2008-03-12 EP claimed
WO-2006137789-A1 Quinoline 3 -sulfonate esters as NK3 receptor modulators ASTRAZENECA AB (SE) 2006-12-28 WO claimed
EP-1896418-A1 QUINOLINE 3 -SULFONATE ESTERS AS NK3 RECEPTOR MODULATORS AstraZeneca AB (SE) 2008-03-12 EP disclosed
WO-2006137789-A1 Quinoline 3 -sulfonate esters as NK3 receptor modulators ASTRAZENECA AB (SE) 2006-12-28 WO disclosed