SCHEMBL4965183

SCHEMBL4965183

COc1ccc2ccc(C=O)c(CN3CCN(C)CC3)c2c1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.50
HTR6 P50406 9/20 0.45
HTR7 P34969 3/20 0.43
HTR1A P08908 2/20 0.43
KDM4E B2RXH2 4/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ALDH1A1 P00352 2/20 0.42
ALOX15 P16050 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
TSHR P16473 1/20 0.41
CHKA P35790 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10471643 0.73 MTNR1A (0.47) ERN1ALDH1A1MAPTTSHR
SCHEMBL1428875 0.72 BCHE (0.57)
SCHEMBL1429039 0.71 AHR (0.49) HTR6KDM4EALDH1A1ALOX15HSD17B10
SCHEMBL14877078 0.71 ALDH1A1 (0.58) ERN1KDM4EALDH1A1HSD17B10MAPT
SCHEMBL15156299 0.70 ALDH1A1 (0.49) KDM4EALDH1A1CHKA
SCHEMBL5506162 0.70 ALDH1A1 (0.56) ERN1KDM4EALDH1A1HSD17B10MAPT
SCHEMBL6413743 0.68 TRIM24 (0.62) ERN1KDM4EALDH1A1HSD17B10MAPT
SCHEMBL1740761 0.68 ERN1 (0.49) ERN1KDM4EL3MBTL1ALDH1A1MAPT
SCHEMBL15475020 0.68 ALDH1A1 (0.54) KDM4EALDH1A1
SCHEMBL4698273 0.67 ALDH1A1 (0.53) ERN1KDM4EL3MBTL1ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957478-A2 NEW COMPOUNDS AstraZeneca AB (SE) 2008-08-20 EP claimed
WO-2007061360-A2 NOVEL 3-BICYCLOCARBONYLAMINOPYRIDINE-2-CARBOXAMIDES OR 3-BICYCLOCARBONYLAMINOPYRAZINE-2-CARBOXAMIDES ASTRAZENECA AB (SE) 2007-05-31 WO claimed