SCHEMBL4965822

SCHEMBL4965822

CCOc1cc(C#N)c(Cc2ccc(CC)cc2)cc1Br

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SNCA P37840 1/20 0.38
ALDH1A1 P00352 2/20 0.38
HSD17B10 Q99714 2/20 0.38
CYP2A6 P11509 1/20 0.37
PDE3B Q13370 2/20 0.36
PDE3A Q14432 2/20 0.36
KDM4E B2RXH2 2/20 0.36
LMNA P02545 2/20 0.36
MAPK1 P28482 1/20 0.36
EGFR P00533 3/20 0.35
ERBB2 P04626 3/20 0.35
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CYP3A4 P08684 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
HPGD P15428 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4969383 0.88 MAOB (0.40) SNCAPDE3BPDE3AEGFRERBB2
SCHEMBL1252946 0.88 SNCA (0.39) SNCAALDH1A1CYP2A6PDE3BPDE3A
SCHEMBL4967384 0.84 SNCA (0.37) SNCAALDH1A1HSD17B10CYP2A6PDE3B
SCHEMBL4969143 0.81 POLB (0.36) SNCACYP2A6PDE3BPDE3ALMNA
SCHEMBL14116545 0.79 MAPT (0.39) ALDH1A1HSD17B10KDM4ELMNAMAPK1
SCHEMBL4967285 0.77 HTR2A (0.46) SNCAPDE3BPDE3AARMAOB
SCHEMBL4967178 0.77 SNCA (0.39) SNCAALDH1A1CYP2A6PDE3BPDE3A
SCHEMBL4966730 0.76 IKBKE (0.36) SLC5A2
SCHEMBL4966718 0.76 IKBKE (0.36) SLC5A2
SCHEMBL4966901 0.76 IKBKE (0.36) SLC5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed