SCHEMBL4967178

SCHEMBL4967178

CCc1ccc(Cc2cc(Br)c(SC)cc2C#N)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SNCA P37840 1/20 0.39
CYP2A6 P11509 1/20 0.38
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
MAOB P27338 2/20 0.35
HPGD P15428 2/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
HIF1A Q16665 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4967204 0.86 MAOB (0.45) SNCAPDE3BPDE3AMAOBHPGD
SCHEMBL4966913 0.80 NPC1 (0.36) ALDH1A1MAPTHIF1AMEN1KMT2A
SCHEMBL1252946 0.78 SNCA (0.39) SNCACYP2A6PDE3BPDE3AMAOB
SCHEMBL4967384 0.77 SNCA (0.37) SNCACYP2A6PDE3BPDE3AALDH1A1
SCHEMBL4965822 0.77 SNCA (0.38) SNCACYP2A6PDE3BPDE3AMAOB
SCHEMBL1250672 0.75 CYP2A6 (0.38) CYP2A6MAOBHPGDALDH1A1MAPT
SCHEMBL4969143 0.72 POLB (0.36) SNCACYP2A6PDE3BPDE3AMAPT
SCHEMBL4965518 0.71 RAB9A (0.40) ALDH1A1MAPTL3MBTL1
SCHEMBL19254702 0.71 CYP2A6 (0.44) CYP2A6MAOBHPGDALDH1A1MAPT
SCHEMBL4967258 0.70 SNCA (0.35) SNCAALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed