SCHEMBL4967285

SCHEMBL4967285

COc1ccc(Cc2cc(Br)c(OC)cc2C#N)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.46
MAOB P27338 1/20 0.44
CNR2 P34972 1/20 0.41
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
SNCA P37840 1/20 0.39
LTA4H P09960 1/20 0.39
AR P10275 4/20 0.39
HTR2C P28335 3/20 0.38
FNTA P49354 1/20 0.38
FNTB P49356 1/20 0.38
PGGT1B P53609 1/20 0.38
TUBB4A P04350 1/20 0.38
TUBB P07437 1/20 0.38
TUBA3C P0DPH7 1/20 0.38
TUBA1B P68363 1/20 0.38
TUBA4A P68366 1/20 0.38
TUBB4B P68371 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4969383 0.90 MAOB (0.40) HTR2AMAOBPDE3BPDE3APOLB
SCHEMBL1252946 0.89 SNCA (0.39) HTR2AMAOBPDE3BPDE3ASNCA
SCHEMBL4969232 0.89 MAOB (0.40) HTR2AMAOBCNR2PDE3BPDE3A
SCHEMBL4967569 0.85 PDE4A (0.39) MAOBAR
SCHEMBL4967204 0.84 MAOB (0.45) HTR2AMAOBPDE3BPDE3APOLB
SCHEMBL4966417 0.80 TBK1 (0.39)
SCHEMBL4969537 0.80 TBK1 (0.39)
SCHEMBL4966426 0.80 TBK1 (0.39)
SCHEMBL181219 0.80 MAOB (0.49) MAOBPDE3BPDE3APOLBGAA
SCHEMBL17278234 0.80 HTR2A (0.50) HTR2ACNR2PDE3BPDE3ALTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed