SCHEMBL4966720

SCHEMBL4966720

CCOc1cccc2c1ccn2Cc1cccc(F)c1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 4/20 0.50
SLC2A1 P11166 1/20 0.48
MAPK14 Q16539 3/20 0.46
DRD2 P14416 1/20 0.46
ALDH1A1 P00352 3/20 0.46
LMNA P02545 3/20 0.46
TDP1 Q9NUW8 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
GRIN1 Q05586 2/20 0.45
GRIN2B Q13224 2/20 0.45
DBH P09172 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
HTT P42858 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
MPO P05164 1/20 0.44
CYP19A1 P11511 2/20 0.43
PDE1A P54750 1/20 0.42
PDE1B Q01064 1/20 0.42
PDE1C Q14123 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3850869 0.77 HTR6 (0.54) HTR6SLC2A1MAPK14ALDH1A1LMNA
SCHEMBL3851817 0.76 HTR6 (0.48) HTR6SLC2A1MAPK14DRD2MPO
SCHEMBL18069184 0.74 HTR6 (0.69) HTR6DRD2
SCHEMBL8685326 0.74 ALDH1A1 (0.72) HTR6SLC2A1ALDH1A1LMNATDP1
SCHEMBL18049242 0.72 HTR6 (0.67) HTR6MAPK14ALDH1A1TDP1SMN1; SMN2
SCHEMBL31258087 0.72 HTR6 (0.55) HTR6SLC2A1ALDH1A1LMNATDP1
SCHEMBL1104768 0.72 HTR6 (0.55) HTR6SLC2A1ALDH1A1LMNATDP1
SCHEMBL12543405 0.71 HTR2C (0.46) HTR6NPSR1
SCHEMBL18045050 0.71 HTR6 (0.43) HTR6LMNAL3MBTL1
Ethoxycarbonyl Group SCHEMBL28763762 0.71 EPHX2 (0.47) SLC2A1ALDH1A1LMNATDP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904483-A1 BENZIMIDAZOLE DERIVATIVES AS 5-HT6,5-HT24 F. Hoffmann-Roche AG (CH) 2008-04-02 EP disclosed
WO-2007006677-A1 BENZIMIDAZOLE DERIVATIVES AS 5-HT6,5-HT24 F. HOFFMANN-LA ROCHE AG (CH) 2007-01-18 WO disclosed