SCHEMBL496675

SCHEMBL496675

Oc1ccc(-c2cnc[nH]2)cc1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 9/20 0.64
ASIC3 Q9UHC3 2/20 0.64
POLB P06746 1/20 0.64
SMN1; SMN2 Q16637 1/20 0.64
CYP3A4 P08684 3/20 0.63
MAPT P10636 1/20 0.55
LTA4H P09960 1/20 0.55
CYP2D6 P10635 2/20 0.52
CYP2E1 P05181 1/20 0.52
CYP2A6 P11509 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2B6 P20813 1/20 0.52
CYP2C19 P33261 1/20 0.52
CYP11B1 P15538 1/20 0.52
CYP11B2 P19099 1/20 0.52
CYP1A2 P05177 1/20 0.50
HPGDS O60760 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17800997 0.86 IDO1 (0.75) IDO1ASIC3POLBSMN1; SMN2CYP3A4
SCHEMBL27880327 0.80 IDO1 (0.67) IDO1ASIC3POLBSMN1; SMN2CYP3A4
SCHEMBL1951516 0.78 IDO1 (1.00) IDO1ASIC3POLBSMN1; SMN2CYP3A4
SCHEMBL205481 0.78 IDO1 (0.64) IDO1ASIC3POLBSMN1; SMN2CYP3A4
SCHEMBL872238 0.78 IDO1 (0.64) IDO1ASIC3POLBSMN1; SMN2CYP3A4
SCHEMBL482297 0.78 IDO1 (0.64) IDO1ASIC3POLBSMN1; SMN2CYP3A4
SCHEMBL14705340 0.78 IDO1 (0.64) IDO1ASIC3POLBSMN1; SMN2CYP3A4
SCHEMBL17782163 0.78 ASIC3 (1.00) IDO1ASIC3POLBSMN1; SMN2CYP3A4
SCHEMBL872388 0.78 POLB (1.00) IDO1ASIC3POLBSMN1; SMN2CYP3A4
SCHEMBL27577902 0.78 IDO1 (0.91) IDO1ASIC3POLBSMN1; SMN2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 120 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE49466-E1 Solution phase homogeneous assays BECKMAN COULTER, INC. (US) 2023-03-21 US claimed
US-10036708-B2 Solution phase homogeneous assays BECKMAN COULTER, INC. (US) 2018-07-31 US claimed
CN-1659278-B Fluorescent detection of peroxidase enzymes LUMIGEN INC 2014-07-09 CN claimed
EP-1509601-B1 FLUORESCENT DETECTION OF PEROXIDASE ENZYMES LUMIGEN INC (US) 2012-12-05 EP claimed
JP-4790905-B2 2011-10-12 JP claimed
US-8012705-B2 Nonseparation assay methods BECKMAN COULTER, INC. (US) 2011-09-06 US claimed
US-20110183361-A1 Nonseparation Assay Methods BECKMAN COULTER, INC. (US) 2011-07-28 US claimed
US-7923213-B2 Nonseparation assay methods BECKMAN COULTER, INC. (US) 2011-04-12 US claimed
US-20100317008-A1 Nonseparation Assay Methods BECKMAN COULTER, INC. (US) 2010-12-16 US claimed
US-20100240070-A1 Nonseparation Assay Methods Using Peroxide Generating Enzymes BECKMAN COULTER, INC. (US) 2010-09-23 US claimed
US-20030232405-A1 Fluorescent detection of peroxidase enzymes LUMIGEN INC. 2003-12-18 US claimed
EP-1019525-A4 CHEMILUMINESCENCE COMPOSITIONS AND METHODS LUMIGEN INC (US) 2003-01-02 EP claimed
EP-0938677-A4 CHEMILUMINESCENT DETECTION METHODS USING DUAL ENZYME-LABELED BINDING PARTNERS LUMIGEN INC (US) 2000-09-27 EP claimed
EP-1019525-A1 CHEMILUMINESCENCE COMPOSITIONS AND METHODS LUMIGEN, INC. (US) 2000-07-19 EP claimed
EP-0938677-A1 CHEMILUMINESCENT DETECTION METHODS USING DUAL ENZYME-LABELED BINDING PARTNERS LUMIGEN, INC. (US) 1999-09-01 EP claimed
US-5922558-A REACTING A PEROXIDASE ENZYME WITH A PEROXIDE AND AT LEAST ONE NOVEL COMPOUND HAVING AN ELECTRON RICH C-C DOUBLE BOND REACTIVE TO PEROXIDASE AND THE PEROXIDE TO PRODUCE AN EXCITED STATE COMPOUND; ALSO USEFUL IN ASSAYS FOR PEROXIDASE ENZYMES LUMIGEN, INC. (US) 1999-07-13 US claimed
WO-1999014358-A1 CHEMILUMINESCENCE COMPOSITIONS AND METHODS LUMIGEN, INC. (US) 1999-03-25 WO claimed
US-5843666-A Chemiluminescent detection methods using dual enzyer-labeled binding partners LUMIGEN, INC. (US) 1998-12-01 US claimed
WO-1998021586-A1 CHEMILUMINESCENT DETECTION METHODS USING DUAL ENZYME-LABELED BINDING PARTNERS LUMIGEN, INC. (US) 1998-05-22 WO claimed
US-5043266-A Immunoassay, reaction between a dihydrophthalazinedione (luminol) and hydrogen peroxide, peroxidase enzyme NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1991-08-27 US claimed