SCHEMBL4966883

SCHEMBL4966883

COC(=O)C1(OCc2ccccc2)CC1.O=C(O)C1(OCc2ccccc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
SLC16A3 O15427 1/20 0.40
SLC16A1 P53985 1/20 0.40
MCTS1 Q9ULC4 1/20 0.40
TACR1 P25103 1/20 0.40
TACR3 P29371 1/20 0.40
ADAM17 P78536 4/20 0.39
DDB1 Q16531 1/20 0.39
CRBN Q96SW2 1/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
SLC1A3 P43003 2/20 0.39
SLC1A2 P43004 2/20 0.39
SLC1A1 P43005 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4033998 0.95 ALDH1A1 (0.44) ALDH1A1TACR1TACR3ADAM17DDB1
SCHEMBL4036434 0.89 KMT2A (0.46) ALDH1A1SLC16A3SLC16A1MCTS1DDB1
SCHEMBL1447732 0.83 CYP2D6 (0.44) ALDH1A1MEN1KMT2ACYP2D6CYP2C9
SCHEMBL5176709 0.82 KMT2A (0.44) ALDH1A1SLC16A3SLC16A1MCTS1DDB1
SCHEMBL26928457 0.80 CYP19A1 (0.44) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL21612946 0.80 MAOB (0.41) ALDH1A1MEN1KMT2ASMN1; SMN2HPGD
SCHEMBL16057453 0.80 KMT2A (0.51) ALDH1A1DDB1CRBNMEN1KMT2A
SCHEMBL4299022 0.78 YAP1 (0.48) TACR1MEN1KMT2A
SCHEMBL31721388 0.78 MEN1 (0.40) ALDH1A1SLC16A3SLC16A1MCTS1MEN1
SCHEMBL27627779 0.78 DDB1 (0.38) ALDH1A1DDB1CRBNMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773780-A4 AMIDO COMPOUNDS AND THEIR USE AS PHARMACEUTICALS INCYTE CORP (US) 2008-01-09 EP disclosed
EP-1773780-A2 AMIDO COMPOUNDS AND THEIR USE AS PHARMACEUTICALS Incyte Corporation (US) 2007-04-18 EP disclosed
WO-2006012227-A2 AMIDO COMPOUNDS AND THEIR USE AS PHARMACEUTICALS INCYTE CORPORATION (US) 2006-02-02 WO disclosed