SCHEMBL4966904

SCHEMBL4966904

COc1ccc(Cc2cc(Br)c(OC3CCOC3)cc2NC(C)=O)cc1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 12/20 0.42
PDE4A P27815 7/20 0.42
PDE4B Q07343 7/20 0.42
PDE4C Q08493 7/20 0.42
SLC5A2 P31639 5/20 0.41
KMT2A Q03164 1/20 0.40
ACACB O00763 2/20 0.38
SLC5A1 P13866 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14116479 1.00 PDE4D (0.42) PDE4DPDE4APDE4BPDE4CSLC5A2
SCHEMBL4966888 1.00 PDE4D (0.42) PDE4DPDE4APDE4BPDE4CSLC5A2
SCHEMBL4967803 0.91 PDE4D (0.40) PDE4DPDE4APDE4BPDE4CSLC5A2
SCHEMBL4967798 0.91 PDE4D (0.40) PDE4DPDE4APDE4BPDE4CSLC5A2
SCHEMBL4969181 0.91 PDE4D (0.40) PDE4DPDE4APDE4BPDE4CSLC5A2
SCHEMBL4965236 0.88 PDE4A (0.45) PDE4DPDE4APDE4BPDE4CKMT2A
SCHEMBL14116724 0.84 PDE4D (0.43) PDE4DPDE4APDE4BPDE4C
SCHEMBL4967553 0.84 PDE4D (0.43) PDE4DPDE4APDE4BPDE4C
SCHEMBL4967561 0.84 PDE4D (0.43) PDE4DPDE4APDE4BPDE4C
SCHEMBL4968389 0.82 ALDH1A1 (0.45) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed