SCHEMBL4969232

SCHEMBL4969232

COc1ccc(Cc2cc(Br)c(OC(C)C)cc2C#N)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.40
HTR2A P28223 1/20 0.37
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
SLC6A4 P31645 2/20 0.36
ESRRA P11474 1/20 0.36
ESR2 Q92731 1/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP2D6 P10635 1/20 0.35
SLC6A2 P23975 1/20 0.35
NOS2 P35228 1/20 0.35
SNCA P37840 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
CNR2 P34972 1/20 0.35
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4967285 0.89 HTR2A (0.46) MAOBHTR2APDE3BPDE3APOLB
SCHEMBL4967384 0.88 SNCA (0.37) PDE3BPDE3ACYP2D6SNCAALDH1A1
SCHEMBL4969383 0.84 MAOB (0.40) MAOBHTR2APDE3BPDE3APOLB
SCHEMBL4967204 0.81 MAOB (0.45) MAOBHTR2APDE3BPDE3AESRRA
SCHEMBL4968294 0.81 HTR2A (0.39) HTR2ASLC6A4CYP2D6ALDH1A1LMNA
SCHEMBL4967569 0.80 PDE4A (0.39) MAOBMEN1KMT2ALMNA
SCHEMBL1252946 0.78 SNCA (0.39) MAOBHTR2APDE3BPDE3AMEN1
SCHEMBL4966426 0.75 TBK1 (0.39) KMT2A
SCHEMBL4969537 0.75 TBK1 (0.39) KMT2A
SCHEMBL4966417 0.75 TBK1 (0.39) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed