SCHEMBL4967340

SCHEMBL4967340

CC(=O)Nc1ccc(Br)c(O[C@@H]2CCOC2)c1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.50
MAPK8 P45983 1/20 0.43
MAPK9 P45984 1/20 0.43
PDE4D Q08499 11/20 0.42
PDE4A P27815 5/20 0.42
PDE4B Q07343 5/20 0.42
PDE4C Q08493 5/20 0.42
ERBB2 P04626 1/20 0.42
EPHA2 P29317 1/20 0.42
KDR P35968 1/20 0.42
EPHB4 P54760 1/20 0.42
GRM4 Q14833 2/20 0.42
STAT1 P42224 1/20 0.42
MAPT P10636 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
PIP5K1C O60331 1/20 0.40
PIK3CA P42336 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4970129 1.00 RORC (0.50) RORCMAPK8MAPK9PDE4DPDE4A
SCHEMBL4967351 1.00 RORC (0.50) RORCMAPK8MAPK9PDE4DPDE4A
SCHEMBL7361005 0.85 PDE4D (0.58) RORCPDE4DPDE4APDE4BPDE4C
SCHEMBL4968732 0.83 RORC (0.59) RORCPDE4DPDE4APDE4BPDE4C
SCHEMBL28446957 0.79 ACACB (0.51) RORCMAPK8MAPK9CYP1A2
SCHEMBL28446956 0.79 ACACB (0.51) RORCMAPK8MAPK9CYP1A2
SCHEMBL22688391 0.79 PDE4D (0.54) PDE4DPDE4APDE4BPDE4C
SCHEMBL4969181 0.74 PDE4D (0.40) MAPK8MAPK9PDE4DPDE4APDE4B
SCHEMBL4967798 0.74 PDE4D (0.40) MAPK8MAPK9PDE4DPDE4APDE4B
SCHEMBL4967803 0.74 PDE4D (0.40) MAPK8MAPK9PDE4DPDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed