SCHEMBL4968181

SCHEMBL4968181

CCc1ccc(Cc2cc(Br)c(OC3CCC3)cc2N)cc1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.38
CSNK2A1 P68400 2/20 0.37
MEN1 O00255 5/20 0.36
KMT2A Q03164 5/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PDE4A P27815 1/20 0.35
NPY1R P25929 1/20 0.35
NPY2R P49146 1/20 0.35
MAPT P10636 1/20 0.35
HRH1 P35367 2/20 0.34
LMNA P02545 1/20 0.34
IKBKB O14920 1/20 0.33
SLC5A1 P13866 2/20 0.33
SLC5A2 P31639 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4967785 0.88 PDE4A (0.41) MEN1KMT2ANPSR1PDE4AMAPT
SCHEMBL4968649 0.86 PDE4D (0.38) PDE4ASLC5A1SLC5A2
SCHEMBL4967734 0.86 PDE4D (0.38) PDE4ASLC5A1SLC5A2
SCHEMBL4967723 0.86 PDE4D (0.38) PDE4ASLC5A1SLC5A2
SCHEMBL4969143 0.81 POLB (0.36) POLBCSNK2A1MEN1KMT2ANPSR1
SCHEMBL1252319 0.81 ALDH1A1 (0.44) POLBMAPTALDH1A1GAA
SCHEMBL14116545 0.80 MAPT (0.39) POLBMEN1KMT2AMAPTLMNA
SCHEMBL4968269 0.78 RORC (0.38) POLBMEN1KMT2ANPSR1IKBKB
SCHEMBL4966698 0.77 CSNK2A1 (0.36) POLBCSNK2A1MEN1KMT2AALDH1A1
SCHEMBL4966210 0.77 KMT2A (0.41) POLBCSNK2A1MEN1KMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed