SCHEMBL4968648

SCHEMBL4968648

Fc1cccc2ccc(C(F)(F)F)nc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKD3 O94806 1/20 0.41
MAP4K4 O95819 1/20 0.41
CDK1 P06493 1/20 0.41
CSF1R P07333 1/20 0.41
PIM1 P11309 1/20 0.41
CDK2 P24941 1/20 0.41
MARK3 P27448 1/20 0.41
AKT1 P31749 1/20 0.41
FLT4 P35916 1/20 0.41
FLT3 P36888 1/20 0.41
FRK P42685 1/20 0.41
MAPKAPK2 P49137 1/20 0.41
CLK2 P49760 1/20 0.41
RPS6KA3 P51812 1/20 0.41
MAPK12 P53778 1/20 0.41
CSNK2A1 P68400 1/20 0.41
CDK5 Q00535 1/20 0.41
MAP4K2 Q12851 1/20 0.41
STK3 Q13188 1/20 0.41
CAMK2D Q13557 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24352377 0.82 AR (0.40) ARLMNAPFKFB3HDAC1HDAC6
SCHEMBL2331355 0.80 TRPV4 (0.41) SLC40A1KDM4ERAB9AP2RX7PTGS2
SCHEMBL3462719 0.80 AURKA (0.41) SRPK1GSK3AGSK3BLMNASLC40A1
SCHEMBL18463777 0.79 AR (0.38) ARLMNAPFKFB3HDAC1HDAC6
SCHEMBL7253959 0.78 METAP2 (0.53) PIM1LMNASMN1; SMN2KDM4ENPC1
SCHEMBL28507492 0.78 MAPT (0.45) SLC40A1KDM4EP2RX7MAPTTDP1
SCHEMBL29496084 0.78 BACE1 (0.53) ARLMNASLC40A1SMN1; SMN2NPC1
SCHEMBL8325687 0.78 ELANE (0.41) ARLMNAPFKFB3SLC40A1PTGS2
SCHEMBL30586432 0.78 ELANE (0.41) ARLMNAPFKFB3SLC40A1PTGS2
SCHEMBL30586451 0.78 MAP4K4 (0.42) MAP4K4CDK2MAPKAPK2RPS6KA3CSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115466212-B 2-trifluoromethyl quinoline compound and synthetic method and application thereof 河南农业大学 2023-09-22 CN disclosed
EP-1968968-A1 COMPOSITIONS AND METHODS FOR MODULATING GATED ION CHANNELS PainCeptor Pharma Corp. (CA) 2008-09-17 EP disclosed
WO-2007071055-A1 COMPOSITIONS AND METHODS FOR MODULATING GATED ION CHANNELS PAINCEPTOR PHARMA CORPORATION (CA) 2007-06-28 WO disclosed
US-4009020-A QUINOLINE-4-CARBOXYLIC ACID OR SALTS AMCHEM PRODUCTS, INC. (US) 1977-02-22 US disclosed