SCHEMBL4968853

SCHEMBL4968853

CCOc1cc(Br)c(Cc2ccc(CC)cc2)cc1I

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.40
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
SLC5A2 P31639 2/20 0.34
CYP3A4 P08684 1/20 0.34
SNCA P37840 1/20 0.34
MAPT P10636 3/20 0.34
HTT P42858 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
KDM4E B2RXH2 1/20 0.34
HPGD P15428 2/20 0.33
POLB P06746 2/20 0.33
ALDH1A1 P00352 1/20 0.33
XBP1 P17861 1/20 0.33
KMT2A Q03164 2/20 0.32
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
RAB9A P51151 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1250647 0.87 HTR2A (0.39) LMNATSHRSLC5A2CYP3A4ALDH1A1
SCHEMBL4965624 0.83 CSNK2A1 (0.33) LMNATSHRCYP3A4SNCAPDE3B
SCHEMBL4966210 0.80 KMT2A (0.41) LMNASLC5A2MAPTPOLBKMT2A
SCHEMBL1252300 0.78 SNCA (0.38) SLC5A2SNCAKMT2APDE3BPDE3A
SCHEMBL4967258 0.78 SNCA (0.35) SNCAMAPTSMN1; SMN2KDM4EPOLB
SCHEMBL4967215 0.77 HSD17B10 (0.47) LMNATSHRHSD17B10MAPTHTT
SCHEMBL27684413 0.76 SMN1; SMN2 (0.44) LMNAMAPTSMN1; SMN2HPGDPOLB
SCHEMBL4967985 0.74 PDE4D (0.38) SLC5A2
SCHEMBL14116528 0.74 PDE4D (0.38) SLC5A2
SCHEMBL14116545 0.73 MAPT (0.39) LMNAHSD17B10SLC5A2CYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed