SCHEMBL4965624

SCHEMBL4965624

CCc1ccc(Cc2cc(I)c(OC(C)C)cc2Br)cc1

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CSNK2A1 P68400 2/20 0.33
SNCA P37840 1/20 0.33
P2RX3 P56373 1/20 0.32
HTR1A P08908 2/20 0.31
HTR2A P28223 2/20 0.31
HTR2C P28335 2/20 0.31
HTR2B P41595 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
TSHR P16473 1/20 0.31
NFKB1 P19838 1/20 0.31
PDE3B Q13370 1/20 0.30
PDE3A Q14432 1/20 0.30
PMP22 Q01453 2/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1250647 0.84 HTR2A (0.39) HTR1AHTR2AHTR2CHTR2BCYP1A2
SCHEMBL4968853 0.83 LMNA (0.40) SNCACYP3A4TSHRPDE3BPDE3A
SCHEMBL4968303 0.78 MAPT (0.41) TSHR
SCHEMBL4966210 0.77 KMT2A (0.41) CSNK2A1LMNA
SCHEMBL1252300 0.76 SNCA (0.38) SNCAPDE3BPDE3A
SCHEMBL4967258 0.75 SNCA (0.35) SNCA
SCHEMBL4966698 0.75 CSNK2A1 (0.36) CSNK2A1P2RX3HTR2AHTR2CHTR2B
SCHEMBL27684413 0.74 SMN1; SMN2 (0.44) HTR2AHTR2CLMNA
SCHEMBL4696889 0.74 CSNK2A1 (0.41) CSNK2A1CYP1A2TSHRLMNA
SCHEMBL4967384 0.72 SNCA (0.37) SNCACYP2D6PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed