SCHEMBL4969191

SCHEMBL4969191

[CH2]C1Cc2cc(F)cc(-c3ccoc3)c2O1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AQP1 P29972 3/20 0.36
DRD2 P14416 1/20 0.32
ALDH1A1 P00352 2/20 0.32
CYP1A2 P05177 2/20 0.32
CYP3A4 P08684 2/20 0.32
CLK4 Q9HAZ1 2/20 0.32
MEN1 O00255 1/20 0.32
CYP2D6 P10635 1/20 0.32
ALOX15 P16050 1/20 0.32
TSHR P16473 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32
HSD17B10 Q99714 1/20 0.32
HTR1A P08908 1/20 0.30
HTR7 P34969 1/20 0.30
GPR84 Q9NQS5 1/20 0.30
PARP1 P09874 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6047930 0.84 DRD2 (0.33) DRD2ALDH1A1CYP1A2CYP3A4CLK4
SCHEMBL4597018 0.83 USP7 (0.37) DRD2ALDH1A1CYP1A2CYP3A4CLK4
SCHEMBL4969196 0.83 PARP1 (0.47) AQP1DRD2ALDH1A1CYP1A2CYP3A4
SCHEMBL4596635 0.82 AQP1 (0.39) AQP1HTR1AHTR7GPR84PARP1
SCHEMBL4225361 0.80 AQP1 (0.58) AQP1DRD2HTR1AHTR7PARP1
SCHEMBL4963747 0.79 AQP1 (0.47) AQP1TSHRHSD17B10PARP1
SCHEMBL4597645 0.79 AQP1 (0.40) AQP1HTR1AHTR7
SCHEMBL4596739 0.79 AQP1 (0.38) AQP1ALDH1A1PARP1
SCHEMBL5060185 0.76 AQP1 (0.40) AQP1CLK4
SCHEMBL4595373 0.76 MAOB (0.38) AQP1DRD2HTR1AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1898895-A2 TREATMENT OF DRUG ABUSE Wyeth (US) 2008-03-19 EP claimed
WO-2006116148-A2 (7-ARLYSUBSTITUTED 2, 3-DIHYDR0-1-BENZ0FURAN-2-YL) ALKYLAMINES IN THE TREATMENT' OF SUBSTANCE ABUSE WYETH (US) 2006-11-02 WO claimed