SCHEMBL4969245

SCHEMBL4969245

O=C(Nc1ccc(OCCN2CCCCC2)cc1)c1ccc2ccccc2c1

nearest known ligand 0.70

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 5/20 0.70
KDR P35968 3/20 0.68
NPC1 O15118 4/20 0.61
RAB9A P51151 4/20 0.61
KMT2A Q03164 2/20 0.61
MEN1 O00255 1/20 0.61
POLB P06746 1/20 0.61
MAPT P10636 1/20 0.61
MCL1 Q07820 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
KDM4E B2RXH2 1/20 0.59
HRH3 Q9Y5N1 1/20 0.58
PSMB1 P20618 2/20 0.58
PSMB5 P28074 2/20 0.58
PSMB2 P49721 1/20 0.58
LTA4H P09960 1/20 0.58
CASP3 P42574 1/20 0.56
SENP7 Q9BQF6 1/20 0.56
GCGR P47871 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL545944 0.83 BRAF (0.53) MCHR1KDRNPC1RAB9AKMT2A
SCHEMBL4968829 0.81 GCGR (0.69) MCHR1KDRNPC1RAB9AKMT2A
SCHEMBL4491205 0.80 HRH3 (0.60) MCHR1KDRNPC1RAB9AKMT2A
SCHEMBL12128447 0.78 HRH4 (0.72) MCHR1KDRNPC1RAB9ASMN1; SMN2
SCHEMBL30186207 0.78 HRH3 (0.81) HRH3LTA4H
SCHEMBL11151279 0.78 HRH3 (0.81) HRH3LTA4H
SCHEMBL14385803 0.77 HRH3 (0.55) MCHR1KDRKDM4EHRH3PSMB1
SCHEMBL5176439 0.77 KDR (0.65) KDRHRH3PSMB1PSMB5LTA4H
SCHEMBL13202486 0.77 HRH3 (0.58) MCHR1KDRKDM4EHRH3
SCHEMBL2112484 0.77 ESR1 (0.61) PSMB1PSMB5PSMB2LTA4HGCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954670-A2 NUCLEAR RECEPTOR BINDING AGENTS GTX Inc. (US) 2008-08-13 EP disclosed
WO-2007062230-A2 NUCLEAR RECEPTOR BINDING AGENTS GTX, INC. (US) 2007-05-31 WO disclosed