SCHEMBL497044

SCHEMBL497044

CCCn1c(C)c(C(=O)c2cccc3ccccc23)c2ccccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 19/20 1.00
CNR1 P21554 9/20 1.00
MEN1 O00255 1/20 1.00
NR1I2 O75469 1/20 1.00
ALDH1A1 P00352 1/20 1.00
CYP1A2 P05177 1/20 1.00
MAPT P10636 1/20 1.00
HPGD P15428 1/20 1.00
TSHR P16473 1/20 1.00
MAPK1 P28482 1/20 1.00
CYP2C19 P33261 1/20 1.00
KMT2A Q03164 1/20 1.00
NR1H4 Q96RI1 1/20 1.00
SLC6A3 Q01959 1/20 0.84

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29989454 0.92 CNR2 (1.00) CNR2CNR1MEN1NR1I2ALDH1A1
SCHEMBL29362163 0.91 CNR2 (1.00) CNR2CNR1MEN1NR1I2ALDH1A1
SCHEMBL16344141 0.91 CNR2 (1.00) CNR2CNR1MEN1NR1I2ALDH1A1
SCHEMBL6324281 0.91 CNR2 (1.00) CNR2CNR1MEN1NR1I2ALDH1A1
SCHEMBL29989324 0.91 CNR2 (1.00) CNR2CNR1MEN1NR1I2ALDH1A1
SCHEMBL9035701 0.90 CNR2 (0.81) CNR2CNR1MEN1NR1I2ALDH1A1
SCHEMBL10093010 0.89 CNR2 (0.81) CNR2CNR1MEN1NR1I2ALDH1A1
SCHEMBL6325870 0.89 CNR2 (1.00) CNR2CNR1MEN1NR1I2ALDH1A1
SCHEMBL29988794 0.89 CNR2 (1.00) CNR2CNR1MEN1NR1I2ALDH1A1
SCHEMBL6330271 0.87 CNR2 (1.00) CNR2CNR1MEN1NR1I2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 295 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4739302-A2 HYALURONIC ACID BASED DRUG DELIVERY SYSTEMS Cella Therapeutics, LLC (US) 2026-05-13 EP claimed
US-20250360137-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES FREEDOM BIOSCIENCES INC (US) 2025-11-27 US claimed
EP-4618980-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES Freedom Biosciences, Inc. (US) 2025-09-24 EP claimed
WO-2025085674-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT OF ULCERATIVE COLITIS BACAINN THERAPEUTICS, INC. (US) 2025-04-24 WO claimed
WO-2025010288-A2 HYALURONIC ACID BASED DRUG DELIVERY SYSTEMS VISUS THERAPEUTICS, INC. (US) 2025-01-09 WO claimed
EP-3664795-B1 CANNABIS AND DERIVATIVES THEREOF FOR THE TREATMENT OF PAIN AND INFLAMMATION RELATED WITH DENTAL PULP AND BONE REGENERATION RELATED TO DENTAL JAW BONE DEFECTS CANNIBITE BVBA (BE) 2024-06-19 EP claimed
WO-2024107445-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES FREEDOM BIOSCIENCES, INC. (US) 2024-05-23 WO claimed
CN-117100863-A Use of cannabinoid systems and downstream pathways thereof for preventing and/or treating chronic itch 南方科技大学 2023-11-24 CN claimed
US-20230181540-A1 COMPOSITIONS AND METHODS FOR ACTIVATING SIGNALING THROUGH THE CB2 CANNABINOID RECEPTOR FOR TREATING AND PREVENTING LYSOSOMAL STORAGE DISEASES AND DISORDERS WYLDER NATION FOUNDATION 2023-06-15 US claimed
EP-4153169-A1 COMPOSITIONS AND METHODS FOR ACTIVATING SIGNALING THROUGH THE CB2 CANNABINOID RECEPTOR FOR TREATING AND PREVENTING LYSOSOMAL STORAGE DISEASES AND DISORDERS Wylder Nation Foundation (US) 2023-03-29 EP claimed
WO-2022204414-A1 FORMULATIONS AND KITS FOR THE DIAGNOSTIC EVALUATION OF INFECTIOUS DISEASES AND METHODS THEREOF VYRIPHARM ENTERPRISES, INC. (US) 2022-09-29 WO claimed
WO-2022204419-A1 SYNTHETIC CANNABINOID COMBINATION THERAPY COMPOSITIONS AND METHODS FOR PERSONALIZED AND TARGETED THERAPIES INCLUDING THE TREATMENT OF INFECTIOUS DISEASES VYRIPHARM ENTERPRISES, INC. (US) 2022-09-29 WO claimed
US-20220305147-A1 SYNTHETIC CANNABINOID COMBINATION THERAPY COMPOSITIONS AND METHODS FOR PERSONALIZED AND TARGETED THERAPIES INCLUDING THE TREATMENT OF INFECTIOUS DISEASES VYRIPHARM ENTERPRISES, INC. 2022-09-29 US claimed
US-20220117932-A1 Lecithin Vesicles CannaClear Inc. (CA) 2022-04-21 US claimed
US-9289421-B2 Methods and compositions for reducing serum levels of immunoglobulin E (IgE) UNIVERSITY OF SOUTH FLORIDA (US) 2016-03-22 US claimed
US-20140350052-A1 Methods and Compositions for Reducing Serum Levels of Immunoglobulin E (IGE) NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2014-11-27 US claimed
WO-2013033155-A1 METHODS AND COMPOSITIONS FOR REDUCING SERUM LEVELS OF IMMUNOGLOBULIN E (IGE) UNIVERSITY OF SOUTH FLORIA (US) 2013-03-07 WO claimed
US-7763607-B2 Pharmaceutical compositions comprising CBx cannabinoid receptor modulators and potassium channel modulators SOLVAY PHARMACEUTICALS GMBH (DE) 2010-07-27 US claimed
US-20060160776-A1 Compositions of a cyclooxygenase-2 selective inhibitor and a cannabinoid agent for the treatment of central nervous system damage PHARMACIA CORPORATION 2006-07-20 US claimed
WO-2004105699-A2 COMPOSITIONS OF A CYCLOOXYGENASE-2 SELECTIVE INHIBITOR AND A CANNABINOID AGENT FOR THE TREATMENT OF CENTRAL NERVOUS SYSTEM DAMAGE PHARMACIA CORPORATION (US) 2004-12-09 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250360137-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES PDE9A, PDE3A, PDE2A CNR2 204/4885CNR1 221/4885MEN1 2211/4885
US-20060160776-A1 Compositions of a cyclooxygenase-2 selective inhibitor and a cannabinoid agent for the treatment of central nervous system damage CNR2, CNR1, PTGS2 CNR2 1/4885CNR1 2/4885MEN1 4616/4885
US-20220305147-A1 SYNTHETIC CANNABINOID COMBINATION THERAPY COMPOSITIONS AND METHODS FOR PERSONALIZED AND TARGETED THERAPIES INCLUDING THE TREATMENT OF INFECTIOUS DISEASES CNR2, CNR1, FAAH CNR2 1/4885CNR1 2/4885MEN1 1926/4885
US-20230181540-A1 COMPOSITIONS AND METHODS FOR ACTIVATING SIGNALING THROUGH THE CB2 CANNABINOID RECEPTOR FOR TREATING AND PREVENTING LYSOSOMAL STORAGE DISEASES AND DISORDERS GBA1, CNR2, CNR1 CNR2 2/4885CNR1 3/4885MEN1 3906/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.