SCHEMBL4970694

SCHEMBL4970694

CC(=O)N1CCN(c2ccc(C(=O)Nc3ccc(Cl)c(Nc4ccccc4F)c3)cn2)CC1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 13/20 0.51
SMO Q99835 1/20 0.49
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
AURKA O14965 1/20 0.47
AURKB Q96GD4 1/20 0.47
KCNQ3 O43525 1/20 0.46
KCNQ2 O43526 1/20 0.46
RAB9A P51151 1/20 0.46
EGFR P00533 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4968074 0.93 SMO (0.52) DGAT1SMOKMT2AAURKAAURKB
SCHEMBL4971826 0.90 SMO (0.50) SMOKMT2ARAB9AEGFR
SCHEMBL4972268 0.89 SMO (0.52) SMOMEN1KMT2AAURKAAURKB
SCHEMBL398151 0.89 SMO (0.53) DGAT1SMOKMT2AAURKAAURKB
SCHEMBL4971048 0.89 RAB9A (0.50) SMOKMT2AAURKAAURKBKCNQ3
SCHEMBL4970651 0.87 SMO (0.51) DGAT1SMOMEN1KMT2AKCNQ3
SCHEMBL4972061 0.87 RAB9A (0.57) SMOKMT2AKCNQ3KCNQ2RAB9A
SCHEMBL402823 0.87 SMO (0.59) SMOMEN1KMT2ARAB9AEGFR
SCHEMBL4971825 0.86 RAB9A (0.54) SMOKMT2ARAB9AEGFR
SCHEMBL403537 0.86 SMO (0.54) SMOKCNQ3KCNQ2RAB9AEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957461-A1 BISAMIDE INHIBITORS OF HEDGEHOG SIGNALING Genentech, Inc. (US) 2008-08-20 EP disclosed
WO-2007059157-A1 BISAMIDE INHIBITORS OF HEDGEHOG SIGNALING GENENTECH, INC. (US) 2007-05-24 WO disclosed