SCHEMBL4968074

SCHEMBL4968074

CC(=O)N1CCN(c2ccc(C(=O)Nc3ccc(Cl)c(Nc4ccccc4Cl)c3)cn2)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 1/20 0.52
MT-CO2 P00403 1/20 0.49
RAB9A P51151 6/20 0.48
DGAT1 O75907 2/20 0.48
EGFR P00533 1/20 0.47
MAPK1 P28482 2/20 0.46
MAPT P10636 2/20 0.46
AURKA O14965 1/20 0.46
AURKB Q96GD4 1/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
USP2 O75604 1/20 0.46
TP53 P04637 1/20 0.46
NPC1 O15118 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
KMT2A Q03164 1/20 0.46
KDM4E B2RXH2 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC3 O15379 1/20 0.44
HDAC2 Q92769 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4971826 0.94 SMO (0.50) SMOMT-CO2RAB9AEGFRMAPK1
SCHEMBL4970694 0.93 DGAT1 (0.51) SMORAB9ADGAT1EGFRAURKA
SCHEMBL4972268 0.93 SMO (0.52) SMORAB9AEGFRMAPK1MAPT
SCHEMBL4972061 0.90 RAB9A (0.57) SMORAB9AEGFRMAPK1MAPT
SCHEMBL402823 0.90 SMO (0.59) SMORAB9AEGFRMAPK1MAPT
SCHEMBL403506 0.89 MAPT (0.56) SMOMT-CO2RAB9AMAPK1MAPT
SCHEMBL4971825 0.89 RAB9A (0.54) SMORAB9AEGFRMAPK1MAPT
SCHEMBL4972451 0.88 SMO (0.58) SMORAB9ADGAT1EGFRMAPK1
SCHEMBL4971048 0.88 RAB9A (0.50) SMORAB9AEGFRMAPK1MAPT
SCHEMBL4971603 0.88 GAA (0.52) SMORAB9ADGAT1EGFRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957461-A1 BISAMIDE INHIBITORS OF HEDGEHOG SIGNALING Genentech, Inc. (US) 2008-08-20 EP claimed
WO-2007059157-A1 BISAMIDE INHIBITORS OF HEDGEHOG SIGNALING GENENTECH, INC. (US) 2007-05-24 WO claimed
EP-1957461-A1 BISAMIDE INHIBITORS OF HEDGEHOG SIGNALING Genentech, Inc. (US) 2008-08-20 EP disclosed
WO-2007059157-A1 BISAMIDE INHIBITORS OF HEDGEHOG SIGNALING GENENTECH, INC. (US) 2007-05-24 WO disclosed