SCHEMBL4972298

SCHEMBL4972298

CC(C)C[C@@](NC(=O)O)(C(=O)N1CCNCC1)C(C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 1/20 0.34
CHRM3 P20309 1/20 0.34
SIGMAR1 Q99720 2/20 0.32
HPGD P15428 1/20 0.31
CA2 P00918 2/20 0.31
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA9 Q16790 1/20 0.31
CHKA P35790 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12308618 0.76 CA2 (0.38) CHRM5CHRM3SIGMAR1HPGDCA2
SCHEMBL22234198 0.74 CA2 (0.39) CHRM3SIGMAR1HPGDCA2CA12
SCHEMBL4972011 0.72 CHRM5 (0.40) CHRM5CHRM3SIGMAR1
SCHEMBL12308679 0.71 CA2 (0.37) CHRM5CHRM3SIGMAR1HPGDCA2
SCHEMBL12308748 0.70 CA2 (0.36) CHRM5CHRM3SIGMAR1HPGDCA2
SCHEMBL22236039 0.69 CA2 (0.42) CHRM5CHRM3SIGMAR1HPGDCA2
SCHEMBL3938238 0.68 CA2 (0.46) CHRM5CHRM3SIGMAR1HPGDCA2
SCHEMBL22233564 0.67 GAA (0.38) SIGMAR1HPGDCA2CA12CA1
SCHEMBL12308783 0.67 GAA (0.38) CHRM5CHRM3SIGMAR1HPGDCA2
SCHEMBL10683 0.66 CA2 (0.48) SIGMAR1HPGDCA2CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968590-A2 NOVEL COMPOUNDS SmithKline Beecham Corporation (US) 2008-09-17 EP disclosed
WO-2007070865-A2 PIPERAZINE COMPOUNDS AS AGONISTS OF TRPV4 CHANNEL RECEPTORS SMITHKLINE BEECHAM CORPORATION (US) 2007-06-21 WO disclosed