SCHEMBL4972011

SCHEMBL4972011

CC(C)C[C@](CN1CCNCC1)(NC(=O)O)C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 1/20 0.40
CHRM3 P20309 1/20 0.40
SIGMAR1 Q99720 3/20 0.38
ALDH1A1 P00352 1/20 0.34
HTT P42858 1/20 0.34
MMP8 P22894 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4971731 0.76 HRH2 (0.33)
SCHEMBL4973854 0.76 SIGMAR1 (0.34) CHRM5CHRM3SIGMAR1ALDH1A1HTT
SCHEMBL4972298 0.72 CHRM5 (0.34) CHRM5CHRM3SIGMAR1
SCHEMBL4595956 0.72 MMP8 (0.39) MMP8
SCHEMBL4596451 0.72 MMP8 (0.39) MMP8
SCHEMBL22235513 0.71 SIGMAR1 (0.41) CHRM5CHRM3SIGMAR1ALDH1A1HTT
SCHEMBL22557833 0.67 SIGMAR1 (0.45) CHRM5CHRM3SIGMAR1ALDH1A1HTT
SCHEMBL5381690 0.66 SIGMAR1 (0.41) CHRM5CHRM3SIGMAR1ALDH1A1HTT
SCHEMBL29057665 0.66 CHRM5 (0.43) CHRM5CHRM3SIGMAR1ALDH1A1MEN1
SCHEMBL2637094 0.64 FFAR1 (0.44) CHRM5CHRM3SIGMAR1ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968590-A2 NOVEL COMPOUNDS SmithKline Beecham Corporation (US) 2008-09-17 EP disclosed
WO-2007070865-A2 PIPERAZINE COMPOUNDS AS AGONISTS OF TRPV4 CHANNEL RECEPTORS SMITHKLINE BEECHAM CORPORATION (US) 2007-06-21 WO disclosed