SCHEMBL4972805

SCHEMBL4972805

C[C@H](COc1ccccc1)N(N)C(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.45
MTNR1A P48039 3/20 0.44
MTNR1B P49286 3/20 0.44
MAOA P21397 1/20 0.42
PTGS1 P23219 1/20 0.42
CYP2D6 P10635 3/20 0.41
ADRB2 P07550 1/20 0.41
ADRB1 P08588 1/20 0.41
ADRB3 P13945 1/20 0.41
ALDH1A1 P00352 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
TSHR P16473 2/20 0.40
SLC22A2 O15244 1/20 0.40
SLC22A1 O15245 1/20 0.40
SLC22A3 O75751 1/20 0.40
ESR1 P03372 1/20 0.40
CHRM2 P08172 1/20 0.40
HTR1A P08908 1/20 0.40
ADRA2A P08913 1/20 0.40
ADORA3 P0DMS8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4972800 1.00 LMNA (0.45) LMNAMTNR1AMTNR1BMAOAPTGS1
SCHEMBL6781747 0.80 ATM (0.44) ADRA2BADRA2CSLC6A2HTR2AADRA1A
SCHEMBL14842276 0.76 HDAC6 (0.33)
SCHEMBL2713474 0.76 HDAC6 (0.33)
SCHEMBL2713471 0.76 HDAC6 (0.33)
SCHEMBL118082 0.75 ALOX5 (0.47) LMNACYP2D6ALDH1A1CYP1A2
SCHEMBL6613322 0.75 ALOX5 (0.47) LMNACYP2D6ALDH1A1CYP1A2
SCHEMBL8771876 0.74 KDM4E (0.41) MTNR1AMTNR1BALDH1A1SMN1; SMN2KDM4E
SCHEMBL28934594 0.74 LMNA (0.50) LMNAMTNR1AMTNR1BMAOAPTGS1
SCHEMBL28934593 0.74 LMNA (0.50) LMNAMTNR1AMTNR1BMAOAPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966139-A1 ASPARTIC PROTEASE INHIBITORS Vitae Pharmaceuticals, Inc. (US) 2008-09-10 EP disclosed
WO-2007070201-A1 ASPARTIC PROTEASE INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2007-06-21 WO disclosed