SCHEMBL4973172

SCHEMBL4973172

Cc1onc(-c2ccccc2)c1-c1c[nH]c(-c2ccc(C(=O)O)cc2)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.48
PTGS1 P23219 4/20 0.48
MAPK14 Q16539 2/20 0.47
KMT2A Q03164 5/20 0.47
GAA P10253 4/20 0.47
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 3/20 0.47
GLA P06280 3/20 0.47
HPGD P15428 3/20 0.47
MEN1 O00255 3/20 0.47
MT-CO2 P00403 3/20 0.45
MAPT P10636 3/20 0.44
NPSR1 Q6W5P4 1/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
LMNA P02545 1/20 0.44
CA3 P07451 1/20 0.44
ADRB2 P07550 1/20 0.44
ADRB1 P08588 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4970984 0.91 GABRA5 (0.46) PTGS2MAPK14KMT2AGAAKDM4E
SCHEMBL2472200 0.89 PTGS2 (0.59) PTGS2PTGS1MAPK14KMT2AGAA
SCHEMBL4973220 0.85 MAPK14 (0.52) MAPK14KMT2AMEN1MAPK8
SCHEMBL4972970 0.84 MAPK14 (0.43) PTGS2PTGS1MAPK14KMT2AALDH1A1
SCHEMBL4971009 0.83 GABRA5 (0.51) MAPK14KMT2AMEN1MAPK8
SCHEMBL4971711 0.83 GABRA5 (0.51) MAPK14KMT2AMEN1MAPK8
SCHEMBL4972650 0.83 KDM4E (0.47) PTGS2PTGS1MAPK14KMT2AGAA
SCHEMBL4973396 0.83 GABRA5 (0.54) MAPK14NPSR1
SCHEMBL4971139 0.82 PTGS2 (0.46) PTGS2PTGS1MAPK14KMT2AGAA
SCHEMBL4973268 0.82 MEN1 (0.49) PTGS2MAPK14KMT2AGAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968973-A2 ARYL-ISOXAZOL-4-YL-IMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2008-09-17 EP disclosed
WO-2007074078-A2 ARYL-ISOXAZOL-4-YL-IMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-07-05 WO disclosed