SCHEMBL4973532

SCHEMBL4973532

C#Cc1cccc(-c2n[c]c3ccncc3n2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 2/20 0.38
CSNK2A2 P19784 2/20 0.35
CSNK2B P67870 2/20 0.35
CSNK2A1 P68400 2/20 0.35
CYP1A2 P05177 7/20 0.35
CYP3A4 P08684 6/20 0.35
CYP2C9 P11712 3/20 0.35
USP2 O75604 2/20 0.35
HPGD P15428 1/20 0.35
CASP1 P29466 1/20 0.35
CLK4 Q9HAZ1 6/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNA5 P30532 1/20 0.34
CHRNA4 P43681 1/20 0.34
ALDH1A1 P00352 6/20 0.34
HSD17B10 Q99714 5/20 0.34
TSHR P16473 4/20 0.34
MAPK1 P28482 4/20 0.34
MEN1 O00255 4/20 0.34
KMT2A Q03164 4/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7662098 0.75 IDO1 (0.42) ABCG2CSNK2A2CSNK2BCSNK2A1CYP1A2
Hydrochloric Acid SCHEMBL7652459 0.74 IDO1 (0.41) ABCG2CSNK2A2CSNK2BCSNK2A1CYP1A2
SCHEMBL8682254 0.69 EGFR (0.43) ABCG2CYP3A4HDAC8LMNA
SCHEMBL28881990 0.69 CYP2A6 (0.56) CYP1A2CYP3A4HPGDCHRNB2CHRNA5
SCHEMBL29984880 0.69 CYP2A6 (0.56) CYP1A2CYP3A4HPGDCHRNB2CHRNA5
SCHEMBL4396963 0.68 CLK4 (0.67) ABCG2CYP1A2CYP3A4CLK4ALDH1A1
SCHEMBL3841296 0.65 CA12 (0.48) ABCG2CYP3A4CYP2C9CLK4MEN1
SCHEMBL22744178 0.65 MAP4K4 (0.37) ABCG2CSNK2A2CSNK2BCSNK2A1CYP1A2
SCHEMBL27819271 0.64 ADORA2A (0.46) ABCG2CYP1A2CYP3A4CYP2C9HPGD
SCHEMBL1801527 0.64 PDGFRB (0.50) CYP1A2HPGDTSHRMAPK1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979348-A2 ANTI-VIRAL COMPOUNDS Abbott Laboratories (US) 2008-10-15 EP disclosed
WO-2007076034-A2 ANTI-VIRAL COMPOUNDS ABBOTT LABORATORIES (US) 2007-07-05 WO disclosed