SCHEMBL4974000

SCHEMBL4974000

Cc1onc(-c2cccc(F)c2)c1CC=O

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 14/20 0.51
THRB P10828 1/20 0.47
ALDH1A1 P00352 3/20 0.46
GPBAR1 Q8TDU6 1/20 0.46
HTR7 P34969 1/20 0.41
PLA2G1B P04054 1/20 0.40
MAPT P10636 1/20 0.40
ATG4B Q9Y4P1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4971798 0.84 ALDH1A1 (0.52) GABRA5ALDH1A1PLA2G1BMAPTATG4B
SCHEMBL4790252 0.83 GABRA5 (0.49) GABRA5THRBALDH1A1
SCHEMBL4723502 0.83 ALDH1A1 (0.56) GABRA5THRBALDH1A1PLA2G1BMAPT
SCHEMBL1777407 0.82 GABRA5 (0.51) GABRA5THRBALDH1A1GPBAR1HTR7
SCHEMBL1777280 0.82 GABRA5 (0.54) GABRA5THRBALDH1A1GPBAR1HTR7
SCHEMBL27814863 0.82 GABRA5 (0.51) GABRA5THRBALDH1A1GPBAR1HTR7
SCHEMBL27814671 0.81 GABRA5 (0.49) GABRA5THRBALDH1A1GPBAR1
SCHEMBL27918192 0.80 GABRA5 (0.55) GABRA5THRBALDH1A1GPBAR1
SCHEMBL21752792 0.80 GABRA5 (0.60) GABRA5ALDH1A1GPBAR1
SCHEMBL21752799 0.79 GPBAR1 (0.48) GABRA5ALDH1A1GPBAR1HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968973-A2 ARYL-ISOXAZOL-4-YL-IMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2008-09-17 EP disclosed
WO-2007074078-A2 ARYL-ISOXAZOL-4-YL-IMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-07-05 WO disclosed