SCHEMBL4975247

SCHEMBL4975247

N#Cc1c(N)cc(Cl)nc1[N+](=O)[O-]

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 5/20 0.38
IKBKB O14920 1/20 0.34
ALDH1A1 P00352 3/20 0.33
TDP1 Q9NUW8 2/20 0.33
GRM6 O15303 1/20 0.33
GRIA1 P42261 1/20 0.33
GRIA2 P42262 1/20 0.33
GRIA3 P42263 1/20 0.33
GRIA4 P48058 1/20 0.33
XDH P47989 1/20 0.33
S1PR4 O95977 1/20 0.33
MAPK1 P28482 1/20 0.33
MAPT P10636 2/20 0.33
HPGD P15428 2/20 0.33
CYP2C9 P11712 2/20 0.33
NPC1 O15118 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
XBP1 P17861 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1629347 0.74 ALDH1A1 (0.42) VCAM1ALDH1A1TDP1GRM6GRIA1
SCHEMBL31288050 0.68 S1PR4 (0.44) ALDH1A1TDP1S1PR4MAPTPOLB
SCHEMBL2307443 0.68 S1PR4 (0.44) ALDH1A1TDP1S1PR4MAPTPOLB
SCHEMBL31569503 0.68 ALDH1A1 (0.40) ALDH1A1TDP1S1PR4MAPTHPGD
SCHEMBL4759212 0.68 VCAM1 (0.49) VCAM1ALDH1A1TDP1GRM6GRIA1
SCHEMBL18462460 0.67 ALDH1A1 (0.47) ALDH1A1TDP1MAPTHPGDNPC1
SCHEMBL29462393 0.67 ALDH1A1 (0.47) ALDH1A1TDP1MAPTHPGDNPC1
SCHEMBL260778 0.67 ALDH1A1 (0.47) ALDH1A1TDP1MAPTHPGDNPC1
SCHEMBL6385999 0.65 ALDH1A1 (0.49) ALDH1A1TDP1MAPK1MAPTNPC1
SCHEMBL3016976 0.65 VCAM1 (0.48) VCAM1ALDH1A1TDP1GRM6GRIA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979351-A1 6-PHENYL-1H-IMIDAZO[4, 5-C]PYRIDINE-4-CARBONITRILE DERIVATIVES AS CATHEPSIN K AND S INHIBITORS N.V. Organon (NL) 2008-10-15 EP disclosed
WO-2007080191-A1 6-PHENYL-1H-IMIDAZO[4, 5-C]PYRIDINE-4-CARBONITRILE DERIVATIVES AS CATHEPSIN K AND S INHIBITORS N.V. ORGANON (NL) 2007-07-19 WO disclosed