SCHEMBL4975853

SCHEMBL4975853

CC1(CCS(=O)(=O)c2ccc(S(C)(=O)=O)cc2)CCN(CC[C@H](c2ccc(S(C)(=O)=O)cc2)c2cc(F)cc(F)c2)CC1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 19/20 0.51
CYP2D6 P10635 1/20 0.51
KCNH2 Q12809 1/20 0.51
CCR2 P41597 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4973495 0.84 CCR5 (0.57) CCR5CYP2D6KCNH2
SCHEMBL5503283 0.82 CCR5 (0.55) CCR5CYP2D6KCNH2CCR2
SCHEMBL3303563 0.81 CCR5 (0.59) CCR5CYP2D6KCNH2
SCHEMBL4977781 0.79 CCR2 (0.46) CCR5CCR2
SCHEMBL5238997 0.77 CCR5 (0.58) CCR5CYP2D6KCNH2CCR2
SCHEMBL4977798 0.76 CCR5 (0.48) CCR5CYP2D6KCNH2
SCHEMBL5502263 0.76 CCR5 (0.48) CCR5CYP2D6KCNH2
SCHEMBL5220283 0.76 CCR5 (0.61) CCR5CYP2D6KCNH2CCR2
SCHEMBL5235987 0.76 CCR5 (0.61) CCR5CYP2D6KCNH2CCR2
SCHEMBL5498416 0.75 CCR5 (0.55) CCR5CYP2D6KCNH2CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080021038-A1 Novel Piperidine/8-Azabicyclo [3.2.1.] Octan Derivatives As Modulators Of Chemokine Receptor Ccr5 TUCKER HOWARD 2008-01-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080021038-A1 Novel Piperidine/8-Azabicyclo [3.2.1.] Octan Derivatives As Modulators Of Chemokine Receptor Ccr5 CCR5, CXCR1, CCR2 CCR5 1/4885CYP2D6 1565/4885KCNH2 1730/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.