SCHEMBL4977322

SCHEMBL4977322

COc1ccc(-c2ccccc2CCN(c2cccnc2)c2cccnc2)c(OC)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
HPGD P15428 1/20 0.38
BRD9 Q9H8M2 1/20 0.37
BRD7 Q9NPI1 1/20 0.37
KCNA5 P22460 2/20 0.34
CYP11B1 P15538 4/20 0.34
CYP11B2 P19099 4/20 0.34
PDE10A Q9Y233 2/20 0.34
RAB9A P51151 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
GAA P10253 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
NPC1 O15118 1/20 0.33
ATM Q13315 1/20 0.33
CYP1A2 P05177 1/20 0.32
METAP2 P50579 1/20 0.32
KCNK3 O14649 1/20 0.32
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL884698 0.75 KCNA5 (0.57) ALDH1A1BRD9BRD7KCNA5RAB9A
SCHEMBL1369604 0.74 BRD9 (0.38) ALDH1A1HPGDBRD9BRD7KCNA5
SCHEMBL4974371 0.74 KCNA5 (0.50) ALDH1A1HPGDKCNA5CYP11B1CYP11B2
SCHEMBL4975470 0.73 KCNA5 (0.51) ALDH1A1KCNA5CYP11B1CYP11B2TSHR
SCHEMBL14536130 0.72 BRD9 (0.52) HPGDBRD9BRD7PDE10AMEN1
SCHEMBL4977357 0.72 GPBAR1 (0.39) CYP11B1CYP11B2CYP1A2CYP2C9
SCHEMBL4975732 0.67 PPARA (0.34) ALDH1A1KCNA5PDE10ATSHRATM
SCHEMBL17276010 0.67 BRD9 (0.56) HPGDBRD9BRD7PDE10ARAB9A
SCHEMBL31438401 0.67 BRD9 (0.56) HPGDBRD9BRD7PDE10ARAB9A
SCHEMBL4979371 0.67 HTR2A (0.44) KCNA5CYP11B1CYP11B2GAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1993551-A2 POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2008-11-26 EP disclosed
WO-2007089735-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2007-08-09 WO disclosed