SCHEMBL4975732

SCHEMBL4975732

C1=C(c2ccccc2CCN(c2cccnc2)c2cccnc2)CCCC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 1/20 0.34
PSMB5 P28074 4/20 0.34
TDP1 Q9NUW8 1/20 0.33
PTGS2 P35354 1/20 0.33
F2RL1 P55085 1/20 0.33
KDR P35968 1/20 0.32
CSF1R P07333 1/20 0.32
ALDH1A1 P00352 2/20 0.31
FFAR2 O15552 1/20 0.31
PIM1 P11309 1/20 0.31
KCNA5 P22460 2/20 0.30
KCNN4 O15554 1/20 0.30
KCNH2 Q12809 1/20 0.30
CHRNB4 P30926 1/20 0.30
CHRNA3 P32297 1/20 0.30
MAPT P10636 1/20 0.30
TSHR P16473 1/20 0.30
HTT P42858 1/20 0.30
ATM Q13315 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4974371 0.77 KCNA5 (0.50) PTGS2ALDH1A1KCNA5KCNH2MAPT
SCHEMBL4975470 0.76 KCNA5 (0.51) ALDH1A1PIM1KCNA5KCNN4KCNH2
SCHEMBL1367820 0.71 F2RL1 (0.40) PPARAPSMB5TDP1PTGS2F2RL1
SCHEMBL4977357 0.70 GPBAR1 (0.39)
SCHEMBL4979371 0.69 HTR2A (0.44) KCNA5KCNN4MAPTTSHRHTT
SCHEMBL22738602 0.67 PTGS2 (0.51) PSMB5TDP1PTGS2FFAR2
SCHEMBL31538073 0.67 PTGS2 (0.48) PSMB5TDP1PTGS2F2RL1
SCHEMBL4977322 0.67 ALDH1A1 (0.38) ALDH1A1KCNA5KCNN4KCNH2TSHR
SCHEMBL3623417 0.66 PDK2 (0.42) ALDH1A1PIM1KCNA5KCNH2L3MBTL1
SCHEMBL1366828 0.66 L3MBTL1 (0.56) ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1993551-A2 POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2008-11-26 EP claimed
WO-2007089735-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2007-08-09 WO claimed