SCHEMBL4979371

SCHEMBL4979371

c1ccc(Cc2ccccc2CCN(c2cccnc2)c2cccnc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.44
CYP11B1 P15538 2/20 0.43
CYP11B2 P19099 2/20 0.43
CHRNA7 P36544 2/20 0.41
HTR1A P08908 1/20 0.40
DRD2 P14416 1/20 0.40
GRM2 Q14416 2/20 0.39
GAA P10253 2/20 0.39
TSHR P16473 1/20 0.39
TBXAS1 P24557 2/20 0.38
HTT P42858 1/20 0.38
KCNA5 P22460 3/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38
KCNN4 O15554 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4974371 0.77 KCNA5 (0.50) CYP11B1CYP11B2TSHRHTTKCNA5
SCHEMBL4975470 0.75 KCNA5 (0.51) CYP11B1CYP11B2CHRNA7TSHRHTT
SCHEMBL1366828 0.73 L3MBTL1 (0.56) MAPK1
SCHEMBL18590701 0.73 GAA (0.53) GRM2GAATSHRKCNA5POLB
SCHEMBL4979253 0.70 CYP11B2 (0.46) CYP11B1CYP11B2KCNA5
SCHEMBL4975773 0.70 KCNA5 (0.39) CYP11B1CYP11B2TSHRKCNA5POLB
SCHEMBL4980305 0.70 KCNA5 (0.39) CYP11B1CYP11B2HTTKCNA5MAPK1
SCHEMBL1367309 0.70 KCNA5 (0.44) CYP11B1CYP11B2GRM2GAATSHR
SCHEMBL4977357 0.70 GPBAR1 (0.39) CYP11B1CYP11B2HTR1ADRD2GRM2
SCHEMBL9129445 0.69 CHRNA7 (0.57) CHRNA7GAAKCNA5KCNN4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1993551-A2 POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2008-11-26 EP claimed
WO-2007089735-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2007-08-09 WO claimed