SCHEMBL4978491

SCHEMBL4978491

Cc1cc(C(=O)N2CCNCC2(Cc2ccccc2)Cc2ccccc2)c(-c2ccccc2)n1-c1cccc(N2CCN(C)CC2)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 3/20 0.35
HTR6 P50406 3/20 0.35
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
TYK2 P29597 1/20 0.35
JAK3 P52333 1/20 0.35
HTR1A P08908 3/20 0.34
HTR7 P34969 2/20 0.34
SLC6A4 P31645 2/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A3 Q01959 1/20 0.34
KIF11 P52732 2/20 0.34
HTR2C P28335 2/20 0.33
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
DRD1 P21728 1/20 0.33
HRH2 P25021 1/20 0.33
HTR1B P28222 1/20 0.33
HTR2A P28223 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4985604 0.79 HTR1A (0.41) HTR6HTR1ASLC6A4SLC6A2SLC6A3
SCHEMBL3493619 0.71 CA1 (0.44) JAK2HTR1AHTR7SLC6A4SLC6A2
SCHEMBL3491841 0.70 HCRTR1 (0.47) SLC6A4SLC6A2SLC6A3KIF11EZH2
SCHEMBL8238486 0.70 HCRTR1 (0.47) NOTUMSLC6A4SLC6A2SLC6A3
SCHEMBL3495194 0.69 CA1 (0.43) JAK2HTR1AHTR7SLC6A4SLC6A2
Hydrochloric Acid SCHEMBL3495897 0.69 HCRTR1 (0.47) NOTUMSLC6A4SLC6A2SLC6A3
SCHEMBL5171411 0.69 CA1 (0.43) JAK2HTR1AHTR7SLC6A4SLC6A2
SCHEMBL8238469 0.69 NOTUM (0.52) NOTUMSIGMAR1ALDH1A1
SCHEMBL8236184 0.66 HCRTR1 (0.53) NOTUMSLC6A4SLC6A2SLC6A3ALDH1A1
Hydrochloric Acid SCHEMBL3494081 0.66 HCRTR1 (0.52) NOTUMSLC6A4SLC6A2SLC6A3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1984355-A2 CYCLIC AMINE COMPOUND AND USE THEREOF FOR THE PROPHYLAXIS OR TREATMENT OF HYPERTENSION Takeda Pharmaceutical Company Limited (JP) 2008-10-29 EP disclosed
WO-2007094513-A2 CYCLIC AMINE COMPOUND AND USE THEREOF FOR THE PROPHYLAXIS OR TREATMENT OF HYPERTENSION TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-08-23 WO disclosed