SCHEMBL4985604

SCHEMBL4985604

Cc1cc(C(=O)N2CCNCC2(Cc2ccccc2)Cc2ccccc2)c(-c2ccccc2)n1-c1ccccc1OCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
HTR6 P50406 4/20 0.41
HIF1A Q16665 2/20 0.40
AVPR2 P30518 1/20 0.39
AVPR1A P37288 1/20 0.39
PTGER1 P34995 3/20 0.38
PARP1 P09874 2/20 0.36
DHODH Q02127 3/20 0.35
SNRNP200 O75643 1/20 0.34
MGLL Q99685 1/20 0.33
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4978491 0.79 NOTUM (0.35) HTR1ASLC6A2SLC6A4SLC6A3HTR6
SCHEMBL3491561 0.78 PTGER1 (0.48) AVPR2AVPR1APTGER1DHODH
SCHEMBL8238361 0.77 MAPT (0.48) AVPR2AVPR1APTGER1DHODH
SCHEMBL3493942 0.74 TSHR (0.47) PTGER1
SCHEMBL3493642 0.71 CA1 (0.45) HIF1AAVPR2AVPR1APTGER1
Hydrochloric Acid SCHEMBL3495368 0.69 HCRTR1 (0.46) SLC6A2SLC6A4SLC6A3
SCHEMBL27573516 0.68 L3MBTL1 (0.43) SLC6A2SLC6A4SLC6A3
SCHEMBL3492269 0.66 HCRTR1 (0.47) SLC6A2SLC6A4SLC6A3HIF1A
SCHEMBL8238469 0.65 NOTUM (0.52)
SCHEMBL4321471 0.65 STS (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1984355-A2 CYCLIC AMINE COMPOUND AND USE THEREOF FOR THE PROPHYLAXIS OR TREATMENT OF HYPERTENSION Takeda Pharmaceutical Company Limited (JP) 2008-10-29 EP disclosed
WO-2007094513-A2 CYCLIC AMINE COMPOUND AND USE THEREOF FOR THE PROPHYLAXIS OR TREATMENT OF HYPERTENSION TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-08-23 WO disclosed