SCHEMBL4983207

SCHEMBL4983207

CCCCc1ccc(N(Cc2ccc(C(C)(C)C)cc2)C(=N)N)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.42
NR1H4 Q96RI1 1/20 0.42
LMNA P02545 1/20 0.41
PTGES O14684 2/20 0.41
ALOX5 P09917 2/20 0.41
STS P08842 2/20 0.38
GRIN2D O15399 1/20 0.37
GRIN3B O60391 1/20 0.37
GRIN1 Q05586 1/20 0.37
GRIN2A Q12879 1/20 0.37
GRIN2B Q13224 1/20 0.37
GRIN2C Q14957 1/20 0.37
GRIN3A Q8TCU5 1/20 0.37
F13A1 P00488 1/20 0.36
TGM2 P21980 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
PLK1 P53350 1/20 0.35
ESRRG P62508 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4985082 0.89 NR1H4 (0.49) KCNH2NR1H4LMNAPTGESALOX5
Hydrochloric Acid SCHEMBL4985557 0.87 NR1H4 (0.48) KCNH2NR1H4LMNAPTGESALOX5
SCHEMBL4981172 0.86 NR1H4 (0.40) NR1H4
Hydrochloric Acid SCHEMBL4981490 0.85 NR1H4 (0.39) NR1H4
SCHEMBL8802180 0.85 ESR1 (0.49) LMNA
SCHEMBL4979785 0.84 TNNC1 (0.41) LMNASTS
SCHEMBL4980138 0.82 NR1H4 (0.44) KCNH2NR1H4LMNAPTGESALOX5
SCHEMBL4994487 0.82 NR1H4 (0.52) KCNH2NR1H4LMNAPTGESALOX5
Hydrochloric Acid SCHEMBL4985726 0.81 NR1H4 (0.43) KCNH2NR1H4LMNAPTGESALOX5
SCHEMBL4981466 0.80 NR1H4 (0.43) NR1H4PTGESALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7351743-B1 Therapeutic guanidines WYETH (US) 2008-04-01 US claimed