SCHEMBL4989442

SCHEMBL4989442

COc1cc(CC2=NCCN2)c(F)cc1NS(C)(=O)=O

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 13/20 0.42
ADRA1D P25100 10/20 0.42
ADRA1B P35368 10/20 0.42
ADRA2A P08913 8/20 0.42
ADRA2C P18825 8/20 0.41
HTR1B P28222 3/20 0.39
ALDH1A1 P00352 2/20 0.36
TAAR1 Q96RJ0 1/20 0.36
HTR1D P28221 2/20 0.36
ADRA2B P18089 1/20 0.36
PTGIR P43119 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4994047 0.90 ADRA1A (0.44) ADRA1AADRA1DADRA1BADRA2AADRA2C
SCHEMBL4989433 0.88 ADRA1A (0.44) ADRA1AADRA1DADRA1BADRA2AADRA2C
SCHEMBL4994677 0.87 ADRA1A (0.47) ADRA1AADRA1DADRA1BADRA2AADRA2C
SCHEMBL4994506 0.84 ADRA1A (0.44) ADRA1AADRA1DADRA1BADRA2AADRA2C
SCHEMBL4986567 0.80 ADRA1A (0.47) ADRA1AADRA1DADRA1BADRA2AADRA2C
SCHEMBL4989586 0.80 ADRA1A (0.42) ADRA1AADRA1DADRA1BADRA2AADRA2C
SCHEMBL4994698 0.80 HTR1B (0.51) ADRA1AADRA1DADRA1BADRA2AADRA2C
SCHEMBL5200788 0.80 HTR1B (0.51) ADRA1AADRA1DADRA1BADRA2AADRA2C
Hydrochloric Acid SCHEMBL5201882 0.79 HTR1B (0.50) ADRA1AADRA1DADRA1BADRA2AADRA2C
SCHEMBL4989420 0.77 KDM4E (0.53) ADRA1AADRA1DADRA1BADRA2AADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6756395-B2 CYCLIZATION OF N-(4-CYANOMETHYLPHENYL)METHANESULFONAMIDES WITH ETHYLENEDIAMINE TO FORM N-(4-IMIDAZOL-2-YLMETHYL)-PHENYL) -METHANESULFONAMIDES; INCONTINENCE, SEXUAL DYSFUNCTION, NASAL CONGESTION, AND CNS DISORDERS; ALPHA 1 ADRENERGIC AGONISTS ROCHE PALO ALTO LLC 2004-06-29 US claimed
US-7407980-B2 Imidazolinylmethyl aralkylsulfonamides ROCHE PALO ALTO LLC (US) 2008-08-05 US disclosed
US-7407980-B2 Imidazolinylmethyl aralkylsulfonamides ROCHE PALO ALTO LLC (US) 2008-08-05 US disclosed
US-7407980-B2 Imidazolinylmethyl aralkylsulfonamides ROCHE PALO ALTO LLC (US) 2008-08-05 US disclosed