SCHEMBL499226

SCHEMBL499226

CN(CCC1(CCCN)NC(=O)c2ccc(Cl)cc21)C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 1/20 0.34
KCNH2 Q12809 2/20 0.32
KIF11 P52732 1/20 0.32
AKR1A1 P14550 1/20 0.32
AKR1B1 P15121 1/20 0.32
CES1 P23141 1/20 0.32
IDO1 P14902 1/20 0.31
PPOX P50336 1/20 0.31
GABRP O00591 1/20 0.31
GABRD O14764 1/20 0.31
GABRA1 P14867 1/20 0.31
GABRB1 P18505 1/20 0.31
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31
GABRA5 P31644 1/20 0.31
GABRA3 P34903 1/20 0.31
GABRA2 P47869 1/20 0.31
GABRB2 P47870 1/20 0.31
GABRA4 P48169 1/20 0.31
GABRE P78334 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL499353 0.90 SLC6A9 (0.35) SLC6A9KCNH2AKR1A1AKR1B1CES1
Trifluoroacetic Acid SCHEMBL499608 0.84 PDK2 (0.37) SLC6A9KCNH2KIF11
Trifluoroacetic Acid SCHEMBL499609 0.84 PDK2 (0.37) SLC6A9KCNH2KIF11
SCHEMBL499980 0.83 HPGD (0.34) SLC6A9AKR1A1AKR1B1IDO1PPOX
SCHEMBL499029 0.77 PDK2 (0.36) SLC6A9
SCHEMBL499028 0.77 PDK2 (0.36) SLC6A9
SCHEMBL8084228 0.70 PDK2 (0.36) SLC6A9CYP3A4
SCHEMBL499153 0.67 SMN1; SMN2 (0.38) CES1IDO1
SCHEMBL499154 0.67 SMN1; SMN2 (0.38) CES1IDO1
SCHEMBL499008 0.65 CES1 (0.35) AKR1A1AKR1B1CES1PPOXKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106221-B2 Renin inhibitors VITAE PHARMACEUTICALS, INC. (US) 2012-01-31 US disclosed
US-20100144825-A1 Renin Inhibitors VITAE PHARMACEUTICALS, INC. 2010-06-10 US disclosed
WO-2008156816-A2 RENIN INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2008-12-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100144825-A1 Renin Inhibitors ACE, REN, DNPEP SLC6A9 1035/4885KCNH2 3262/4885KIF11 2932/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.