SCHEMBL4993274

SCHEMBL4993274

CC(C)(C)c1[c]ccc(OCCCCO)c1C(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 1/20 0.36
LOX P28300 1/20 0.33
AOC3 Q16853 1/20 0.33
RARA P10276 1/20 0.31
RARB P10826 1/20 0.31
RARG P13631 1/20 0.31
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL459472 0.73 CA12 (0.31)
SCHEMBL4989706 0.71 TSHR (0.42) ALDH1A1KDM4E
SCHEMBL8725705 0.68 LOX (0.36) ALDH1A1KDM4ELOXAOC3HSD17B10
SCHEMBL248878 0.67 CNR2 (0.46) ALDH1A1LOXAOC3HSD17B10
SCHEMBL11006202 0.65 ALDH1A1 (0.73) ALDH1A1KDM4EHSD17B10
SCHEMBL30292271 0.64 KDM4E (0.47) ALDH1A1KDM4EHSD17B10
SCHEMBL9935540 0.64 TUBB1 (0.33) ALDH1A1
SCHEMBL14200178 0.62 KDM4E (0.49) ALDH1A1KDM4E
SCHEMBL2139323 0.62
SCHEMBL9592076 0.61 SMN1; SMN2 (0.54) ALDH1A1KDM4EAOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080214660-A1 Compounds and Methods for the Inhibition of the Expression of VCAM-1 CRABTREE ACQUISITION CO, LLC 2008-09-04 US disclosed
US-7375252-B2 Compounds and method for the inhibition of the expression of VCAM-1 ATHEROGENICS, INC. (US) 2008-05-20 US disclosed
US-7189870-B2 Compounds and methods for the inhibition of the expression of VCAM-1 ATHEROGENIC, INC. (US) 2007-03-13 US disclosed
US-20050090487-A1 Compounds and methods for the inhibition of the expression of VCAM-1 ATHEROGENICS, INC. 2005-04-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080214660-A1 Compounds and Methods for the Inhibition of the Expression of VCAM-1 VCAM1, ICAM1, SELL ALDH1A1 100/4885KDM4E 2945/4885LOX 242/4885
US-20050090487-A1 Compounds and methods for the inhibition of the expression of VCAM-1 VCAM1, ICAM1, SELL ALDH1A1 100/4885KDM4E 2945/4885LOX 242/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.