SCHEMBL4994516

SCHEMBL4994516

COc1c(N)ccc(CC2=NCCN2)c1C

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 9/20 0.57
HTR1B P28222 8/20 0.57
ADRA2A P08913 4/20 0.49
ADRA2B P18089 4/20 0.49
ADRA2C P18825 4/20 0.49
ADRA1A P35348 4/20 0.49
ADRA1D P25100 3/20 0.49
ADRA1B P35368 3/20 0.49
TAAR1 Q96RJ0 6/20 0.46
PTGIR P43119 1/20 0.44
LMNA P02545 2/20 0.43
CYP2D6 P10635 2/20 0.43
MAPK1 P28482 2/20 0.43
HTR1A P08908 1/20 0.43
MAPT P10636 1/20 0.43
OPRM1 P35372 1/20 0.43
NISCH Q9Y2I1 1/20 0.43
CYP1A2 P05177 1/20 0.42
TSHR P16473 1/20 0.42
RAD52 P43351 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4994510 0.82 HTR1B (0.53) HTR1DHTR1BADRA2AADRA2BADRA2C
SCHEMBL4993062 0.82 HTR1D (0.58) HTR1DHTR1BADRA2AADRA2BADRA2C
SCHEMBL4990257 0.82 HTR1D (0.58) HTR1DHTR1BADRA2AADRA2BADRA2C
SCHEMBL4993251 0.78 HTR1B (0.48) HTR1DHTR1BADRA2AADRA2BADRA2C
SCHEMBL14092041 0.77 HTR1D (0.47) HTR1DHTR1BADRA2AADRA2BADRA2C
SCHEMBL957285 0.75 HTR1D (0.73) HTR1DHTR1BADRA2AADRA2BADRA2C
Bromide SCHEMBL959007 0.74 HTR1D (0.71) HTR1DHTR1BADRA2AADRA2BADRA2C
SCHEMBL953395 0.73 TAAR1 (0.55) HTR1DHTR1BADRA2AADRA2BADRA2C
SCHEMBL4992378 0.73 ALDH1A1 (0.61) HTR1DHTR1BADRA2AADRA2BADRA2C
SCHEMBL10934485 0.73 HTR1B (0.53) HTR1DHTR1BADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7407980-B2 Imidazolinylmethyl aralkylsulfonamides ROCHE PALO ALTO LLC (US) 2008-08-05 US disclosed