SCHEMBL5007455

SCHEMBL5007455

CC1=C(c2ccc(S(C)(=O)=O)cc2)S(=O)(=O)NC12CCCCC2

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 18/20 0.43
PTGS1 P23219 6/20 0.43
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
BRD4 O60885 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5001155 0.82 PTGS2 (0.37) PTGS2PTGS1BRD4
SCHEMBL5007425 0.80 GALR1 (0.36) PTGS2PTGS1KMT2ABRD4
SCHEMBL4994770 0.78 PTGS2 (0.34) PTGS2PTGS1BRD4
SCHEMBL5963380 0.72 GALR1 (0.40) KMT2ASMN1; SMN2
SCHEMBL5963597 0.69 GALR1 (0.38) SMN1; SMN2
SCHEMBL5964141 0.69 GRIA2 (0.36)
SCHEMBL8384211 0.64 PTGS2 (0.88) PTGS2PTGS1
SCHEMBL12341698 0.62 PTGS2 (0.68) PTGS2PTGS1
SCHEMBL5963305 0.62 SLC6A3 (0.39)
SCHEMBL6994135 0.62 PTGS2 (0.43) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7396846-B2 Growth hormone secretagogues ELI LILLY AND COMPANY (US) 2008-07-08 US disclosed
US-7396846-B2 Growth hormone secretagogues ELI LILLY AND COMPANY (US) 2008-07-08 US disclosed
US-7396846-B2 Growth hormone secretagogues ELI LILLY AND COMPANY (US) 2008-07-08 US disclosed
US-20050240001-A1 2-(2-Amino-2-methylpropionylamino)-3-(2,6-difluoro-3-methylphenyl)methoxy propionic acid N-[5-(4-chlorophenyl)-3,3-dimethyl-1,1-dioxo-2,3-dihydroisothiazol-4-ylmethyl]-N-ethylamide; endogenous human growth hormone controller; non-peptidyl in nature, more metabolically stable ELI LILLY AND COMPANY (US) 2005-10-27 US disclosed