SCHEMBL5011863

SCHEMBL5011863

CC(=O)C1(C2(C#N)CC2)C=CC(c2ccccc2)C(F)=C1

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
CACNA1D Q01668 1/20 0.32
POLB P06746 1/20 0.31
CTSC P53634 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5013488 0.76 KDM1A (0.30) KDM4EALDH1A1MAPTKMT2A
SCHEMBL1222086 0.67 EDNRA (0.33) CACNA1D
SCHEMBL6694686 0.64 CACNA1D (0.30) CACNA1D
SCHEMBL4178861 0.60 PPARG (0.35)
SCHEMBL6679649 0.59 CACNA1D (0.35) ALDH1A1CACNA1DPOLB
SCHEMBL9842403 0.58 ELANE (0.33)
SCHEMBL9842547 0.58 CACNA1D (0.33) CACNA1D
SCHEMBL6682470 0.58 TSHR (0.36) KDM4EMEN1ALDH1A1KMT2ACACNA1D
SCHEMBL8393880 0.57 CACNA1D (0.30) CACNA1D
SCHEMBL16534046 0.57

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893562-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B Merck Frosst Canada Ltd. (CA) 2008-03-05 EP disclosed
WO-2006133559-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B MERCK FROSST CANADA LTD. (CA) 2006-12-21 WO disclosed