SCHEMBL5012155

SCHEMBL5012155

CC1CN(c2c(F)cc(-c3csnn3)cc2C=O)CC(C)O1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.34
HTT P42858 1/20 0.34
PDE3B Q13370 2/20 0.34
PDE3A Q14432 2/20 0.34
GAK O14976 2/20 0.33
HPGD P15428 2/20 0.32
CYP2C19 P33261 2/20 0.32
ALDH1A1 P00352 3/20 0.31
KMT2A Q03164 2/20 0.31
MEN1 O00255 1/20 0.31
ERN1 O75460 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP2C9 P11712 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
POLB P06746 1/20 0.30
NOTUM Q6P988 1/20 0.30
MET P08581 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5012752 0.83 KDM4E (0.34) KDM4EHTTGAKHPGDCYP2C19
SCHEMBL4508573 0.78 KDM4E (0.42) KDM4EHTTPDE3BPDE3AERN1
SCHEMBL5015663 0.78 GSK3B (0.36) KDM4EHTTPDE3BPDE3AGAK
SCHEMBL3075477 0.74 KDM4E (0.39) KDM4EHTTPDE3BPDE3AALDH1A1
SCHEMBL4505828 0.74 HTT (0.39) KDM4EHTTPDE3BPDE3AALDH1A1
SCHEMBL3066876 0.71 KDM4E (0.36) KDM4EHTTPDE3BPDE3AALDH1A1
SCHEMBL12726451 0.71 TSHR (0.38) KDM4EHTTHPGDALDH1A1KMT2A
SCHEMBL12703780 0.71 TSHR (0.38) KDM4EHTTHPGDALDH1A1KMT2A
SCHEMBL15609918 0.71 ALDH1A1 (0.38) KDM4EHTTPDE3BPDE3AHPGD
SCHEMBL3070590 0.70 KDM4E (0.37) KDM4EHTTPDE3BPDE3AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888597-A2 ANTIBACTERIAL AGENTS Warner-Lambert Company LLC (US) 2008-02-20 EP disclosed
WO-2006120563-A2 ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY LLC (US) 2006-11-16 WO disclosed