SCHEMBL5015663

SCHEMBL5015663

Cc1nnc(-c2cc(F)c(N3CC(C)OC(C)C3)c(C=O)c2)s1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 7/20 0.36
DYRK1A Q13627 7/20 0.36
WNT1 P04628 3/20 0.36
KDM4E B2RXH2 2/20 0.34
HTT P42858 1/20 0.34
PDE3B Q13370 2/20 0.34
PDE3A Q14432 2/20 0.34
ALDH1A1 P00352 3/20 0.32
ERN1 O75460 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
GAA P10253 2/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
LMNA P02545 1/20 0.32
GAK O14976 2/20 0.31
FFAR4 Q5NUL3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5011046 0.83 KDM4E (0.34) KDM4EHTTALDH1A1GAAL3MBTL1
SCHEMBL5012158 0.83 KDM4E (0.34) KDM4EHTTALDH1A1GAAL3MBTL1
SCHEMBL5011042 0.83 KDM4E (0.34) KDM4EHTTALDH1A1GAAL3MBTL1
SCHEMBL5014296 0.80 KDM4E (0.33) KDM4EHTTALDH1A1
SCHEMBL3069764 0.79 KDM4E (0.34) KDM4EHTT
SCHEMBL3065399 0.79 KDM4E (0.34) KDM4EHTT
SCHEMBL2216534 0.79 GSK3B (0.36) GSK3BDYRK1AWNT1ALDH1A1CYP1A2
SCHEMBL5012250 0.79 GAK (0.32) KDM4EHTTGAK
SCHEMBL5012155 0.78 KDM4E (0.34) KDM4EHTTPDE3BPDE3AALDH1A1
SCHEMBL2258284 0.75 L3MBTL1 (0.36) KDM4EHTTALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888597-A2 ANTIBACTERIAL AGENTS Warner-Lambert Company LLC (US) 2008-02-20 EP disclosed
WO-2006120563-A2 ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY LLC (US) 2006-11-16 WO disclosed