SCHEMBL5013370

SCHEMBL5013370

COCCCCc1cccc2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.46
CYP2C19 P33261 2/20 0.46
CYP2D6 P10635 1/20 0.46
AKR1B1 P15121 1/20 0.46
SIGMAR1 Q99720 1/20 0.46
NQO2 P16083 1/20 0.45
GPR84 Q9NQS5 1/20 0.44
CYP2C9 P11712 1/20 0.44
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
ACP3 P15309 1/20 0.43
MTNR1A P48039 1/20 0.43
IP6K1 Q92551 1/20 0.43
CDYL Q9Y232 1/20 0.43
ATM Q13315 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2092988 0.98 CYP1A2 (0.44) CYP1A2CYP2C19CYP2D6AKR1B1SIGMAR1
SCHEMBL2094194 0.95 CYP1A2 (0.47) CYP1A2CYP2C19CYP2D6AKR1B1SIGMAR1
SCHEMBL791971 0.87 CYP1A2 (0.50) CYP1A2CYP2C19CYP2D6AKR1B1NQO2
SCHEMBL30487942 0.87 CYP1A2 (0.50) CYP1A2CYP2C19CYP2D6AKR1B1NQO2
SCHEMBL9800436 0.84 CYP1A2 (0.58) CYP1A2CYP2C19CYP2D6SIGMAR1NQO2
SCHEMBL5013367 0.82 NQO2 (0.45) CYP1A2CYP2C19CYP2D6SIGMAR1NQO2
SCHEMBL27645176 0.81 BCHE (0.49) SIGMAR1CYP2C9MTNR1ACDYL
SCHEMBL2092985 0.81 NQO2 (0.44) CYP1A2CYP2C19CYP2D6SIGMAR1NQO2
SCHEMBL5830948 0.80 GPR84 (0.59) CYP1A2CYP2C19CYP2D6SIGMAR1NQO2
SCHEMBL460016 0.79 BCHE (0.52) CYP1A2CYP2C19CYP2D6SIGMAR1NQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678185-B1 2,3-DIHYDRO-6-NITROIMIDAZO [2,1-B] OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMA CO LTD (JP) 2008-10-08 EP disclosed
EP-1678185-A1 2,3-DIHYDRO-6-NITROIMIDAZO [2,1-B] OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-07-12 EP disclosed
WO-2005042542-A1 2,3-DIHYDRO-6-NITROIMIDAZO (2,1-B) OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2005-05-12 WO disclosed