SCHEMBL5013584

SCHEMBL5013584

OC(c1ccc(-c2ccc(CC(O)(F)F)cc2)cc1)C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.36
ESR2 Q92731 3/20 0.36
CYP4F2 P78329 1/20 0.35
CYP4A11 Q02928 1/20 0.35
NR1I2 O75469 1/20 0.35
CTSK P43235 2/20 0.34
KIF11 P52732 1/20 0.33
KDM5B Q9UGL1 1/20 0.32
PTPN5 P54829 1/20 0.32
RORC P51449 1/20 0.31
APP P05067 1/20 0.31
CETP P11597 1/20 0.31
FFAR1 O14842 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28043083 0.81 NR1I2 (0.41) ESR1ESR2CYP4F2CYP4A11NR1I2
SCHEMBL13974407 0.80 TSHR (0.41) ESR1ESR2CYP4F2CYP4A11NR1I2
SCHEMBL12323306 0.77 ESR1 (0.42) ESR1ESR2CYP4F2CYP4A11NR1I2
SCHEMBL14593355 0.76 ESR1 (0.48) ESR1ESR2CYP4F2CYP4A11NR1I2
SCHEMBL4497165 0.75 KIF11 (0.46) NR1I2KIF11PTPN5APP
SCHEMBL8988146 0.75 ESR1 (0.58) ESR1ESR2KIF11
SCHEMBL12628146 0.75 KIF11 (0.46) NR1I2KIF11PTPN5APP
SCHEMBL5865851 0.73 TSHR (0.45) ESR1ESR2CYP4F2CYP4A11NR1I2
SCHEMBL5013479 0.73 ESR1 (0.39) ESR1ESR2KIF11RORC
SCHEMBL7370695 0.73 LOXL2 (0.43) ESR1ESR2CYP4F2CYP4A11NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893562-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B Merck Frosst Canada Ltd. (CA) 2008-03-05 EP claimed
WO-2006133559-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B MERCK FROSST CANADA LTD. (CA) 2006-12-21 WO claimed